SCHEMBL15775264

SCHEMBL15775264

Nc1ccc(-c2cc3ncccc3c(=O)[nH]2)cc1

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 1/20 0.52
PARP1 P09874 10/20 0.51
TNKS O95271 6/20 0.51
TNKS2 Q9H2K2 5/20 0.51
ADORA2A P29274 2/20 0.44
ADORA1 P30542 2/20 0.44
ACVR1 Q04771 1/20 0.41
AURKA O14965 2/20 0.41
QTRT1 Q9BXR0 1/20 0.41
KDM4E B2RXH2 1/20 0.40
NPC1 O15118 1/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
HPGD P15428 1/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
AURKB Q96GD4 1/20 0.40
PARP2 Q9UGN5 1/20 0.40
PARP3 Q9Y6F1 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8602417 0.86 ADORA2A (0.59) PARP1TNKSTNKS2ADORA2AADORA1
SCHEMBL15775722 0.85 CCNB2 (0.55) RIPK1PARP1TNKSTNKS2ADORA2A
SCHEMBL15775696 0.85 TNKS (0.57) PARP1TNKSTNKS2ADORA2AADORA1
SCHEMBL15775268 0.85 CCNB2 (0.55) PARP1TNKSTNKS2ADORA2AADORA1
SCHEMBL15775563 0.85 PARP1 (0.56) PARP1TNKSTNKS2ADORA2AADORA1
SCHEMBL15775369 0.82 TNKS (0.59) PARP1TNKSTNKS2ADORA2AADORA1
SCHEMBL4773542 0.82 PARP1 (0.59) RIPK1PARP1TNKSTNKS2KDM4E
SCHEMBL12385912 0.78 PARP1 (0.51) RIPK1PARP1TNKSTNKS2AURKA
SCHEMBL13495429 0.77 PIK3CD (0.53) PARP1TNKSTNKS2ACVR1PARP2
SCHEMBL348483 0.76 PTGER3 (0.47) PARP1TNKSTNKS2ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014087165-A1 TANKYRASE INHIBITORS UNIVERSITY OF BATH (GB) 2014-06-12 WO disclosed