SCHEMBL1586483

SCHEMBL1586483

O=C(O)c1c[nH]c(=O)c(Cc2ccc(F)c(F)c2)c1

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DAO P14920 4/20 0.44
KDM5A P29375 2/20 0.40
KDM5B Q9UGL1 2/20 0.40
ALDH1A1 P00352 1/20 0.37
TSHR P16473 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
PARP1 P09874 1/20 0.37
NOTUM Q6P988 1/20 0.37
VNN1 O95497 1/20 0.36
RXRA P19793 1/20 0.36
PPARA Q07869 1/20 0.36
MAOA P21397 1/20 0.35
MAOB P27338 1/20 0.35
MPO P05164 1/20 0.35
KDM4C Q9H3R0 1/20 0.35
KLKB1 P03952 1/20 0.35
KLK1 P06870 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16881058 0.83 PTPN1 (0.35) DAOTSHRRXRAKDM4CKLKB1
SCHEMBL14604111 0.81 GAA (0.45) DAOTSHRNOTUM
SCHEMBL6471052 0.81 RNASEH1 (0.47) KDM5AKDM5BTSHR
SCHEMBL7268031 0.80 SRD5A2 (0.54) DAOKDM5AKDM5BALDH1A1RXRA
SCHEMBL16486420 0.78 TSHR (0.43) DAOTSHRNOTUMKDM4C
SCHEMBL4649050 0.77 PNP (0.42) DAOALDH1A1L3MBTL1NOTUM
SCHEMBL3344960 0.77 PTPN5 (0.47) DAO
SCHEMBL4381378 0.75 DAO (0.40) DAOKDM5AKDM5BALDH1A1TSHR
SCHEMBL16880522 0.75 KMT2A (0.56) ALDH1A1NOTUMKLKB1KLK1
SCHEMBL16880471 0.75 NAPRT (0.39) DAOPARP1NOTUMRXRAKDM4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2490687-A1 COMPOSITIONS FOR TREATMENT OF CYSTIC FIBROSIS AND OTHER CHRONIC DISEASES Vertex Pharmaceuticals Incorporated (US) 2012-08-29 EP disclosed
WO-2011050325-A1 COMPOSITIONS FOR TREATMENT OF CYSTIC FIBROSIS AND OTHER CHRONIC DISEASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-04-28 WO disclosed
EP-2231280-A2 ORGANIC COMPOUNDS Novartis AG (CH) 2010-09-29 EP disclosed
WO-2009074575-A2 ORGANIC COMPOUNDS NOVARTIS AG (CH) 2009-06-18 WO disclosed