SCHEMBL4649050

SCHEMBL4649050

O=C(O)c1c[nH]c(=O)c(Cc2ccncc2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PNP P00491 1/20 0.42
DAO P14920 1/20 0.42
NAPRT Q6XQN6 1/20 0.42
MAPK7 Q13164 2/20 0.40
HDAC1 Q13547 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
ITK Q08881 2/20 0.39
AURKA O14965 1/20 0.39
TTK P33981 1/20 0.39
AURKB Q96GD4 1/20 0.39
INCENP Q9NQS7 1/20 0.39
NOTUM Q6P988 1/20 0.39
LMNA P02545 2/20 0.38
ALDH1A1 P00352 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
CYP17A1 P05093 1/20 0.38
PLA2G7 Q13093 1/20 0.38
PDE3B Q13370 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14604111 0.86 GAA (0.45) DAONOTUMMEN1KMT2APDE3B
SCHEMBL7268031 0.82 SRD5A2 (0.54) DAOALDH1A1MEN1KMT2A
SCHEMBL16486420 0.80 TSHR (0.43) DAONAPRTNOTUMKMT2A
SCHEMBL3344960 0.79 PTPN5 (0.47) DAOLMNA
SCHEMBL6471052 0.77 RNASEH1 (0.47) PNP
SCHEMBL1586483 0.77 DAO (0.44) DAONOTUMALDH1A1L3MBTL1
SCHEMBL16880522 0.77 KMT2A (0.56) HDAC1HDAC6NOTUMALDH1A1KMT2A
SCHEMBL4649823 0.76 KDM4E (0.45) PNPDAOALDH1A1L3MBTL1
SCHEMBL7432519 0.75 DAO (0.42) PNPDAOMEN1KMT2APDE3B
SCHEMBL6209517 0.74 NOTUM (0.53) DAONOTUMALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1960367-A2 SUBSTITUTED PYRAZOLE COMPOUNDS USEFUL AS SOLUBLE EPOXIDE HYDROLASE INHIBITORS Boehringer Ingelheim International GmbH (DE) 2008-08-27 EP disclosed
WO-2007067836-A2 SUBSTITUTED PYRAZOLE COMPOUNDS USEFUL AS SOLUBLE EPOXIDE HYDROLASE INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-06-14 WO disclosed