SCHEMBL15865262

SCHEMBL15865262

CC(C)c1[nH]nnc1-c1cc(-c2ccc(F)c(CN3CCOCC3)c2)cnc1N

nearest known ligand 0.64

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 14/20 0.64
AXL P30530 1/20 0.39
MERTK Q12866 1/20 0.39
ALOX5AP P20292 2/20 0.39
FEN1 P39748 2/20 0.39
KCNH2 Q12809 1/20 0.38
MET P08581 1/20 0.37
ALK Q9UM73 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19086091 0.88 LRRK2 (0.64) LRRK2KCNH2
SCHEMBL19086093 0.82 LRRK2 (0.64) LRRK2
SCHEMBL15865279 0.81 LRRK2 (0.59) LRRK2ALOX5APFEN1KCNH2MET
SCHEMBL15865510 0.80 LRRK2 (0.65) LRRK2ALOX5APFEN1KCNH2MET
SCHEMBL15864797 0.78 LRRK2 (1.00) LRRK2
SCHEMBL15864772 0.76 LRRK2 (0.64) LRRK2KCNH2MET
SCHEMBL15864661 0.75 LRRK2 (0.65) LRRK2KCNH2MET
SCHEMBL15865168 0.75 LRRK2 (0.65) LRRK2KCNH2MET
SCHEMBL15864658 0.73 LRRK2 (0.66) LRRK2AXLMERTKKCNH2MET
SCHEMBL15864636 0.73 LRRK2 (0.48) LRRK2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2941425-A1 AMINOPYRIDINE DERIVED COMPOUNDS AS LRRK2 INHIBITORS H. Lundbeck A/S (DK) 2015-11-11 EP disclosed
WO-2014106612-A1 AMINOPYRIDINE DERIVED COMPOUNDS AS LRRK2 INHIBITORS H. LUNDBECK A/S (DK) 2014-07-10 WO disclosed