SCHEMBL15904641

SCHEMBL15904641

COc1cnc2cc(-c3ccncc3)[nH]c2c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNB2 O95067 3/20 0.48
CDK1 P06493 3/20 0.48
CCNB1 P14635 3/20 0.48
GSK3A P49840 3/20 0.48
GSK3B P49841 3/20 0.48
CCNB3 Q8WWL7 3/20 0.48
CDK5 Q00535 2/20 0.48
CDK5R1 Q15078 2/20 0.48
PDGFRB P09619 4/20 0.47
PDGFRA P16234 4/20 0.47
KDM4E B2RXH2 2/20 0.45
MAPT P10636 2/20 0.45
MEN1 O00255 1/20 0.45
ALDH1A1 P00352 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
HPGD P15428 1/20 0.45
ALOX15 P16050 1/20 0.45
MAPK1 P28482 1/20 0.45
CASP1 P29466 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17840915 0.77 TGFBR1 (0.53) GSK3B
SCHEMBL15058354 0.73 KDM4E (0.72) CCNB2CDK1CCNB1CCNB3PDGFRB
SCHEMBL16729146 0.73 AXL (0.44) CCNB2CDK1CCNB1GSK3BCCNB3
SCHEMBL21812461 0.71 CYP11B1 (0.56) CDK5CDK5R1KDM4EMAPTMEN1
SCHEMBL2289799 0.71 DAO (0.47) CCNB2CDK1CCNB1GSK3AGSK3B
SCHEMBL21643937 0.70 NPC1 (0.54) GSK3AGSK3BPDGFRBPDGFRAKDM4E
SCHEMBL15904794 0.70 NTRK1 (0.48) GSK3BCDK5CDK5R1MAPK1HSD17B10
SCHEMBL1374700 0.69 MMP12 (0.47) KDM4EALDH1A1CYP1A2CYP3A4HPGD
SCHEMBL25723819 0.69 CYP1A2 (0.38) KDM4EMAPTMEN1ALDH1A1CYP1A2
SCHEMBL4782250 0.69 KDM4E (0.63) CCNB2CDK1CCNB1GSK3AGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014115071-A1 KINASE INHIBITORS CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2014-07-31 WO claimed
WO-2014115071-A1 KINASE INHIBITORS CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2014-07-31 WO disclosed