SCHEMBL15911575

SCHEMBL15911575

CC1CN(c2ccccc2-c2cnc(N3CCC(O)CC3)nc2)CCN1C(C=O)n1ccc2ccncc21

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.37
HCRTR2 O43614 7/20 0.32
HCRTR1 O43613 5/20 0.32
AOC3 Q16853 3/20 0.32
JAK2 O60674 1/20 0.32
JAK3 P52333 1/20 0.32
WDR5 P61964 3/20 0.32
SMO Q99835 1/20 0.31
CXCR3 P49682 2/20 0.31
KCNH2 Q12809 2/20 0.31
TNK2 Q07912 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15911260 0.88 WDR5 (0.36) MAPTHCRTR2WDR5
SCHEMBL15911410 0.87 SMO (0.35) HCRTR2HCRTR1AOC3WDR5SMO
SCHEMBL169439 0.78 CXCR3 (0.52) MAPTHCRTR2HCRTR1CXCR3KCNH2
SCHEMBL15911219 0.78 MAPT (0.38) MAPTHCRTR2HCRTR1AOC3WDR5
SCHEMBL15911272 0.77 WDR5 (0.36) WDR5SMOCXCR3KCNH2
SCHEMBL115607 0.74 HTR1A (0.37) MAPTKCNH2
SCHEMBL114031 0.72 CXCR3 (0.35) CXCR3
SCHEMBL165747 0.70 CXCR3 (0.49) HCRTR2HCRTR1CXCR3KCNH2
SCHEMBL165509 0.68 CXCR3 (0.51) CXCR3KCNH2
SCHEMBL114718 0.67 CXCR3 (0.39) AOC3SMOCXCR3KCNH2TNK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2424840-B1 CXCR3 RECEPTOR ANTAGONISTS BOEHRINGER INGELHEIM INT (DE) 2014-08-06 EP disclosed