SCHEMBL15918600

SCHEMBL15918600

Cc1ccnc(OCC(F)F)c1F

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ACACB O00763 4/20 0.35
CYP17A1 P05093 1/20 0.34
HCRTR1 O43613 4/20 0.33
HCRTR2 O43614 4/20 0.33
DRD1 P21728 1/20 0.33
MKNK2 Q9HBH9 2/20 0.33
CCR1 P32246 1/20 0.31
CCR5 P51681 1/20 0.31
CCR8 P51685 1/20 0.31
MBOAT4 Q96T53 1/20 0.31
NOS3 P29474 3/20 0.31
NOS2 P35228 3/20 0.31
SCN9A Q15858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12903576 0.79 HPGD (0.47) DRD1CCR1CCR5CCR8NOS3
SCHEMBL23624004 0.77 CCR1 (0.38) DRD1CCR1CCR5CCR8NOS3
SCHEMBL11194894 0.75 ADRB1 (0.54)
SCHEMBL31068654 0.71 ACACB (0.32) ACACBHCRTR1HCRTR2
SCHEMBL23990294 0.69 UHRF1 (0.42) HCRTR1HCRTR2CCR1CCR5CCR8
SCHEMBL22308085 0.67 CCR1 (0.37) CCR1CCR5CCR8NOS3NOS2
SCHEMBL16012007 0.67 LOXL2 (0.41)
Ammonia Solution, Strong SCHEMBL28411378 0.67 CYP17A1 (0.50) CYP17A1
SCHEMBL22842968 0.67 HCRTR2 (0.37) HCRTR1HCRTR2MKNK2
SCHEMBL28033606 0.67 TRPA1 (0.47) ACACBNOS3NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014114578-A1 PYRROLIDINE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS AND USES THEREOF BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-07-31 WO disclosed