SCHEMBL15919375

SCHEMBL15919375

CC(C)(C)OC(=O)NCC(=O)Nc1cc(-c2ccc(C#Cc3ccc(CN4CCOCC4)cc3)cc2)nc2ccncc12

nearest known ligand 0.45

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MOK Q9UQ07 13/20 0.45
ACP1 P24666 3/20 0.44
KCNH2 Q12809 1/20 0.40
PDE10A Q9Y233 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15919372 0.86 MOK (0.54) MOKACP1KCNH2PDE10A
SCHEMBL15905202 0.76 KCNH2 (0.52) MOKACP1KCNH2
SCHEMBL15919371 0.75 ACP1 (0.46) MOKACP1KCNH2
SCHEMBL30422422 0.72 TSHR (0.53)
SCHEMBL15919445 0.72 MAPT (0.48) MOK
SCHEMBL30834312 0.70 MOK (0.66) MOK
SCHEMBL15919600 0.70 KCNH2 (0.56) MOKACP1KCNH2
SCHEMBL15919351 0.69 MEN1 (0.45) ACP1
SCHEMBL30834329 0.69 MOK (0.64) MOK
SCHEMBL3713512 0.69 TBK1 (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9663488-B2 Metalloenzyme inhibitor compounds VIAMET PHARMACEUTICALS, INC. (US) 2017-05-30 US disclosed
US-9663488-B2 Metalloenzyme inhibitor compounds VIAMET PHARMACEUTICALS, INC. (US) 2017-05-30 US disclosed
US-20150353546-A1 METALLOENZYME INHIBITOR COMPOUNDS Viamet Pharmaceuticals (NC), Inc. 2015-12-10 US disclosed
US-20150353546-A1 METALLOENZYME INHIBITOR COMPOUNDS Viamet Pharmaceuticals (NC), Inc. 2015-12-10 US disclosed
WO-2014117090-A1 METALLOENZYME INHIBITOR COMPOUNDS VIAMET PHARMACEUTICALS, INC. (US) 2014-07-31 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150353546-A1 METALLOENZYME INHIBITOR COMPOUNDS MMEL1, GPX1, MPO MOK 4173/4885ACP1 2825/4885KCNH2 2250/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.