SCHEMBL15925264

SCHEMBL15925264

Cc1ccnc2nc(N3CCN(C)CC3)cnc12

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 7/20 0.50
HTR3A P46098 3/20 0.50
HRH3 Q9Y5N1 1/20 0.48
TLR9 Q9NR96 5/20 0.44
MET P08581 2/20 0.44
ALDH1A1 P00352 3/20 0.43
CYP1A2 P05177 3/20 0.43
CYP2D6 P10635 2/20 0.43
HSD17B10 Q99714 2/20 0.43
HTR3E A5X5Y0 1/20 0.43
HTR3B O95264 1/20 0.43
HTR3D Q70Z44 1/20 0.43
HTR3C Q8WXA8 1/20 0.43
CYP3A4 P08684 1/20 0.43
TSHR P16473 1/20 0.43
CLK4 Q9HAZ1 1/20 0.43
USP2 O75604 1/20 0.41
ALOX15 P16050 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15925256 0.84 ALDH1A1 (0.43) ALDH1A1CYP1A2HSD17B10TSHRCLK4
SCHEMBL23333325 0.73 CCR1 (0.40) ALDH1A1CYP1A2
SCHEMBL14029975 0.69 HRH4 (0.67) HRH4HTR3AHRH3ALDH1A1CYP1A2
SCHEMBL23332993 0.67 NOS2 (0.41)
SCHEMBL12847495 0.67 CCR1 (0.38)
SCHEMBL14237709 0.67 TLR9 (0.64) HRH4HTR3ATLR9MET
SCHEMBL14237703 0.67 TLR9 (0.64) HRH4HTR3ATLR9METALDH1A1
SCHEMBL27904291 0.67 HRH4 (0.53) HRH4HTR3AHRH3METALDH1A1
SCHEMBL606857 0.67 HRH4 (1.00) HRH4HTR3AHRH3METALDH1A1
SCHEMBL81828 0.67 HTR3A (0.52) HRH4HTR3AHRH3HTR3EHTR3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2229391-B1 PYRIDO[2,3-B]PYRAZINE-8-SUBSTITUTED COMPOUNDS AND THEIR USE CANCER REC TECH LTD (GB) 2014-08-06 EP disclosed