SCHEMBL15948359

SCHEMBL15948359

Nc1nncc(-c2ccc(F)c(-c3ccccc3)c2C(F)(F)F)n1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.39
HSD17B10 Q99714 1/20 0.39
ADORA2A P29274 9/20 0.38
ADORA1 P30542 9/20 0.38
ATR Q13535 2/20 0.36
USP7 Q93009 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.33
CYP11B2 P19099 1/20 0.33
FEN1 P39748 3/20 0.32
ALOX5AP P20292 2/20 0.32
POLB P06746 1/20 0.32
ADORA2B P29275 1/20 0.32
HTR1B P28222 1/20 0.32
HTR2B P41595 1/20 0.32
GPR65 Q8IYL9 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15948360 0.80 KDM4E (0.39) KDM4EHSD17B10ADORA2AADORA1ATR
SCHEMBL3395736 0.72 ADORA2A (0.50) KDM4EHSD17B10ADORA2AADORA1ATR
SCHEMBL31018102 0.72 MPL (0.50) KDM4EADORA2AADORA1ATRL3MBTL1
SCHEMBL2324805 0.72 MPL (0.50) KDM4EADORA2AADORA1ATRL3MBTL1
SCHEMBL2325695 0.71 ADORA2A (0.67) KDM4EHSD17B10ADORA2AADORA1L3MBTL1
SCHEMBL31009002 0.71 ADORA2A (0.67) KDM4EHSD17B10ADORA2AADORA1L3MBTL1
SCHEMBL3128136 0.71 ATR (0.48) ADORA2AADORA1ATRFEN1ALOX5AP
SCHEMBL3399237 0.68 ADORA2A (0.68) KDM4EHSD17B10ADORA2AADORA1L3MBTL1
SCHEMBL2323758 0.66 ADORA2A (0.44) ADORA2AADORA1L3MBTL1CYP11B2FEN1
SCHEMBL2320341 0.66 ADORA2A (0.44) KDM4EADORA2AADORA1L3MBTL1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8809525-B2 1,2,4-triazine-4-amine derivatives HEPTARES THERAPEUTICS LIMITED (GB) 2014-08-19 US disclosed