SCHEMBL3128136

SCHEMBL3128136

Nc1nncc(-c2ccccc2C(F)(F)F)n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATR Q13535 2/20 0.48
PTPN1 P18031 4/20 0.45
NOTUM Q6P988 1/20 0.44
HSD11B1 P28845 1/20 0.42
ADORA2A P29274 1/20 0.42
ADORA1 P30542 1/20 0.42
KMO O15229 1/20 0.41
BACE1 P56817 1/20 0.41
TLR8 Q9NR97 1/20 0.41
MPL P40238 1/20 0.40
CDC7 O00311 1/20 0.40
CCNE1 P24864 1/20 0.40
CDK2 P24941 1/20 0.40
DBF4 Q9UBU7 1/20 0.40
ALOX5AP P20292 1/20 0.40
FEN1 P39748 1/20 0.40
ACP1 P24666 1/20 0.40
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CNR2 P34972 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3248212 0.81 NOTUM (0.44) ATRNOTUMHSD11B1KMOACP1
SCHEMBL3395686 0.79 HSD17B1 (0.40) ATRADORA2AADORA1ALOX5APFEN1
SCHEMBL2324805 0.78 MPL (0.50) ATRNOTUMADORA2AADORA1MPL
SCHEMBL31018102 0.78 MPL (0.50) ATRNOTUMADORA2AADORA1MPL
SCHEMBL28008349 0.77 NOTUM (0.44) ATRPTPN1NOTUMHSD11B1KMO
SCHEMBL5918379 0.77 TRPV1 (0.42) ADORA2AADORA1
SCHEMBL3398117 0.77 MPL (0.44) HSD11B1ADORA2AADORA1MPLALOX5AP
SCHEMBL15948360 0.77 KDM4E (0.39) ATRADORA2AADORA1MPLALOX5AP
SCHEMBL3396593 0.76 KDM4E (0.45) ADORA2AADORA1
SCHEMBL3394338 0.76 AR (0.41) ATRADORA2AADORA1ACP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010046780-A2 ANTI VIRAL COMPOUNDS INSTITUT PASTEUR KOREA (KR) 2010-04-29 WO disclosed
WO-2010046780-A2 ANTI VIRAL COMPOUNDS INSTITUT PASTEUR KOREA (KR) 2010-04-29 WO disclosed
WO-2010001220-A1 NEW 1,2,4-TRIAZINE DERIVATIVES AND BIOLOGICAL APPLICATIONS THEREOF MUTABILIS SA (FR) 2010-01-07 WO disclosed
EP-2141164-A1 New 1,2,4-triazine derivatives and biological applications thereof Mutabilis (FR) 2010-01-06 EP disclosed