SCHEMBL15949025

SCHEMBL15949025

CCS(=O)(=O)c1ccc(-c2ccc(C(CC(=O)c3ccncc3)c3ccccc3)cc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.42
PLOD2 O00469 1/20 0.42
PLOD3 O60568 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
HPGD P15428 1/20 0.42
CYP2C19 P33261 1/20 0.42
PLOD1 Q02809 1/20 0.42
HIF1A Q16665 1/20 0.42
RORC P51449 2/20 0.42
RPS6KA5 O75582 4/20 0.41
AKT1 P31749 4/20 0.41
GSK3B P49841 4/20 0.41
PRKCD Q05655 4/20 0.41
PRKG2 Q13237 4/20 0.41
ROCK1 Q13464 4/20 0.41
PRKG1 Q13976 4/20 0.41
PKN2 Q16513 4/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15949098 0.89 ALDH1A1 (0.43) ALDH1A1PLOD2PLOD3CYP1A2CYP3A4
SCHEMBL362642 0.85 GPBAR1 (0.61) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL369688 0.85 GPBAR1 (0.61) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL369687 0.85 GPBAR1 (0.61) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL15949170 0.81 CYP17A1 (0.44) ALDH1A1RORCNPC1RAB9ASMN1; SMN2
SCHEMBL15949140 0.81 CTSS (0.46) RORC
SCHEMBL369594 0.81 ALDH1A1 (0.61) ALDH1A1PLOD2PLOD3CYP1A2CYP3A4
SCHEMBL15949109 0.80 HPGD (0.46) ALDH1A1PLOD2PLOD3CYP1A2CYP3A4
SCHEMBL15949141 0.80 PLOD2 (0.46) ALDH1A1PLOD2PLOD3CYP1A2CYP3A4
SCHEMBL15949055 0.78 GPBAR1 (0.48) ALDH1A1PLOD2PLOD3CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-B1 1-HYDROXYIMINO-3-PHENYL-PROPANES HOFFMANN LA ROCHE (CH) 2014-08-20 EP claimed