SCHEMBL15958710

SCHEMBL15958710

CC(=O)NC(CO)(CO)CCc1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.46
NPC1 O15118 1/20 0.44
MAPT P10636 1/20 0.44
RAB9A P51151 1/20 0.44
RECQL P46063 2/20 0.43
SSTR4 P31391 1/20 0.43
THRB P10828 1/20 0.42
TAAR1 Q96RJ0 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.41
POLB P06746 1/20 0.41
HPGD P15428 1/20 0.41
MMP8 P22894 1/20 0.40
KEAP1 Q14145 1/20 0.40
HDAC2 Q92769 2/20 0.40
HDAC8 Q9BY41 2/20 0.40
HDAC6 Q9UBN7 2/20 0.40
KDM4E B2RXH2 2/20 0.40
TDP1 Q9NUW8 1/20 0.39
HDAC3 O15379 1/20 0.39
HDAC4 P56524 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16202271 0.94 LMNA (0.46) ALDH1A1NPC1MAPTRAB9ARECQL
SCHEMBL8495637 0.90 POLB (0.45) ALDH1A1NPC1MAPTRAB9ARECQL
SCHEMBL1497771 0.87 FFAR1 (0.53) ALDH1A1NPC1MAPTRAB9ASMN1; SMN2
SCHEMBL9891052 0.85 S1PR1 (0.42) ALDH1A1NPC1RAB9ATAAR1KDM4E
SCHEMBL17427772 0.85 PLK1 (0.44) ALDH1A1THRBPOLBKDM4E
SCHEMBL24430171 0.85 NPC1 (0.45) ALDH1A1NPC1RAB9ASMN1; SMN2HPGD
SCHEMBL5992356 0.84 DPP4 (0.54) NPC1MAPTRAB9ATHRBHDAC2
SCHEMBL8496037 0.84 S1PR1 (0.52) ALDH1A1NPC1MAPTRAB9ATAAR1
SCHEMBL588956 0.84 POLB (0.42) NPC1MAPTTAAR1SMN1; SMN2POLB
SCHEMBL7614431 0.83 ALDH1A1 (0.40) ALDH1A1NPC1MAPTRAB9ARECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111087357-B Preparation method of Prisamod 中国医学科学院药物研究所 2022-07-19 CN disclosed
CN-111087356-B Preparation method of Iguratimod 中国医学科学院药物研究所 2022-06-21 CN disclosed
US-20220153684-A1 PROCESS FOR PREPARATION OF FINGOLIMOD HYDROCHLORIDE SHIVALIK RASAYAN LIMITED (IN) 2022-05-19 US disclosed
CN-111087356-A Preparation method of Iguratimod 中国医学科学院药物研究所 2020-05-01 CN disclosed
CN-111087357-A Preparation method of Prisamod 中国医学科学院药物研究所 2020-05-01 CN disclosed
US-9133096-B2 Process for the production of 2-amino-2[2-(4-C2-20-alkyl-phenyl)ethyl]propane-1,3-diols, and to compounds for use therein NOVARTIS AG (CH) 2015-09-15 US disclosed
EP-2268603-B1 PROCESS FOR THE PREPARATION OF 2-AMINO-2- [2- (4-C3-C21-ALKYL-PHENYL)ETHYL]PROPANE-1, 3-DIOLS NOVARTIS AG (CH) 2015-04-22 EP disclosed
US-8809571-B2 Process for the production of 2-amino-2-[2-(4-C2-20-alkyl-phenyl)ethyl]propane-1,3-diols, and to compounds for use therein NOVARTIS AG (CH) 2014-08-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220153684-A1 PROCESS FOR PREPARATION OF FINGOLIMOD HYDROCHLORIDE S1PR2, S1PR4, S1PR5 ALDH1A1 1249/4885NPC1 1348/4885MAPT 2344/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.