SCHEMBL15966536

SCHEMBL15966536

COC(=O)C(CCN(Cc1ccccc1)Cc1ccccc1)N(COC(C)=O)C(=O)OC

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.42
EPOR P19235 2/20 0.41
ALDH1A1 P00352 2/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
LMNA P02545 1/20 0.39
POLB P06746 1/20 0.39
HSD17B10 Q99714 1/20 0.39
KMT2A Q03164 2/20 0.37
DPP7 Q9UHL4 1/20 0.37
MEN1 O00255 1/20 0.37
HDAC3 O15379 2/20 0.37
HDAC1 Q13547 2/20 0.37
HDAC2 Q92769 2/20 0.37
HDAC8 Q9BY41 2/20 0.37
NCOR2 Q9Y618 2/20 0.37
CHRNB2 P17787 1/20 0.37
CHRNB4 P30926 1/20 0.37
CHRNA3 P32297 1/20 0.37
CHRNA4 P43681 1/20 0.37
HCRTR2 O43614 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15966571 1.00 TSHR (0.42) TSHREPORALDH1A1L3MBTL1LMNA
SCHEMBL17350549 0.76 ABCB1 (0.39) TSHREPORALDH1A1L3MBTL1LMNA
SCHEMBL2456291 0.72 KMT2A (0.48) EPORALDH1A1L3MBTL1LMNAPOLB
SCHEMBL3223085 0.71 TSHR (0.69) TSHRALDH1A1L3MBTL1LMNAPOLB
SCHEMBL27655077 0.71 ALDH1A1 (0.47) TSHRALDH1A1L3MBTL1LMNAPOLB
SCHEMBL7023844 0.70 CASR (0.43) TSHRALDH1A1L3MBTL1LMNAKMT2A
SCHEMBL25181400 0.69 EPOR (0.52) EPORALDH1A1L3MBTL1LMNAPOLB
SCHEMBL12671106 0.68 TSHR (0.65) TSHRALDH1A1LMNAPOLBKMT2A
SCHEMBL13434071 0.68 KMT2A (0.70) ALDH1A1L3MBTL1LMNAPOLBHSD17B10
SCHEMBL24991861 0.66 EPOR (0.58) EPORALDH1A1L3MBTL1LMNAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2957555-A1 METHOD FOR MODIFYING DERIVATIVES OF AMINO ACIDS AND PEPTIDES, COMPOUNDS PRODUCED, AND USE Consejo Superior De Investigaciones Científicas (CSIC) (ES) 2015-12-23 EP disclosed
WO-2014125145-A1 METHOD FOR MODIFYING DERIVATIVES OF AMINO ACIDS AND PEPTIDES, COMPOUNDS PRODUCED, AND USE CONSEJO SUPERIOR DE INVESTIGACIONES CIENTÍFICAS (CSIC) (ES) 2014-08-21 WO disclosed