SCHEMBL17350549

SCHEMBL17350549

COC(=O)C[C@@H](CN(Cc1ccccc1)Cc1ccccc1)N(COC(C)=O)C(=O)OC

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 2/20 0.39
ALDH1A1 P00352 2/20 0.38
POLB P06746 2/20 0.38
LMNA P02545 1/20 0.38
HSD17B10 Q99714 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
MAOB P27338 1/20 0.38
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
TSHR P16473 1/20 0.36
CTRB1 P17538 1/20 0.34
CHRNB2 P17787 1/20 0.34
CHRNB4 P30926 1/20 0.34
CHRNA3 P32297 1/20 0.34
CHRNA4 P43681 1/20 0.34
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
KCNA5 P22460 1/20 0.33
NR1H3 Q13133 1/20 0.32
RORC P51449 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15966536 0.76 TSHR (0.42) ALDH1A1POLBLMNAHSD17B10L3MBTL1
SCHEMBL15966571 0.76 TSHR (0.42) ALDH1A1POLBLMNAHSD17B10L3MBTL1
SCHEMBL27655077 0.75 ALDH1A1 (0.47) ALDH1A1POLBLMNAL3MBTL1TSHR
SCHEMBL24766843 0.73 MEN1 (0.46) ABCB1ALDH1A1POLBLMNAL3MBTL1
SCHEMBL22100562 0.73 MEN1 (0.46) ABCB1ALDH1A1POLBLMNAL3MBTL1
SCHEMBL3450839 0.71 MEN1 (0.41) ABCB1ALDH1A1POLBLMNAL3MBTL1
SCHEMBL3450837 0.71 MEN1 (0.41) ABCB1ALDH1A1POLBLMNAL3MBTL1
SCHEMBL14085934 0.70 MEN1 (0.43) ABCB1ALDH1A1POLBLMNAMAOB
SCHEMBL13657503 0.68 MAOB (0.45) ABCB1ALDH1A1POLBLMNAHSD17B10
SCHEMBL3364898 0.68 NPC1 (0.52) ALDH1A1POLBLMNAL3MBTL1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2957555-A1 METHOD FOR MODIFYING DERIVATIVES OF AMINO ACIDS AND PEPTIDES, COMPOUNDS PRODUCED, AND USE Consejo Superior De Investigaciones Científicas (CSIC) (ES) 2015-12-23 EP disclosed