SCHEMBL15975129

SCHEMBL15975129

COc1ccc2c(Cc3cccc(-c4noc(=O)[nH]4)n3)c(C3CCCCC3)[nH]c2c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 1/20 0.41
MTNR1B P49286 1/20 0.41
PDE10A Q9Y233 3/20 0.39
AGTR1 P30556 3/20 0.35
ALDH1A1 P00352 3/20 0.35
KDM4E B2RXH2 2/20 0.35
RAB9A P51151 1/20 0.35
GAA P10253 1/20 0.34
HPGD P15428 1/20 0.34
ALOX15 P16050 1/20 0.34
CASP1 P29466 1/20 0.34
HTT P42858 1/20 0.34
CASP7 P55210 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HSD17B10 Q99714 1/20 0.34
ALPL P05186 1/20 0.34
CYP1A2 P05177 1/20 0.33
CYP2E1 P05181 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C8 P10632 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15975093 0.83 PDE10A (0.42) PDE10AALDH1A1KDM4ERAB9AHPGD
SCHEMBL15975194 0.83 PDE10A (0.40) PDE10AALDH1A1KDM4EHPGDSMN1; SMN2
SCHEMBL11978656 0.82 PDE10A (0.44) MTNR1AMTNR1BPDE10AALDH1A1KDM4E
SCHEMBL15975094 0.80 CYP19A1 (0.47) PDE10AALDH1A1CASP1HSD17B10USP2
SCHEMBL15975112 0.79 MTNR1A (0.40) MTNR1AMTNR1BPDE10AALDH1A1KDM4E
SCHEMBL11978281 0.79 TUBB4A (0.42) PDE10AAGTR1ALDH1A1KDM4EHSD17B10
SCHEMBL4568577 0.79 MTNR1A (0.48) MTNR1AMTNR1BALDH1A1KDM4EHPGD
SCHEMBL4568450 0.78 MTNR1A (0.50) MTNR1AMTNR1BALDH1A1KDM4EGAA
SCHEMBL4568574 0.78 MTNR1A (0.47) MTNR1AMTNR1BALDH1A1KDM4EHPGD
SCHEMBL4568448 0.77 MTNR1A (0.48) MTNR1AMTNR1BALDH1A1KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8815903-B2 Indole derivative and pharmacologically acceptable salt thereof KISSEI PHARMACEUTICAL CO., LTD. (JP) 2014-08-26 US disclosed
US-8815903-B2 Indole derivative and pharmacologically acceptable salt thereof KISSEI PHARMACEUTICAL CO., LTD. (JP) 2014-08-26 US disclosed