SCHEMBL15975112

SCHEMBL15975112

COc1ccc2c(Cc3cccc(C4=NNNN4)n3)c(C3CCCCC3)[nH]c2c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 1/20 0.40
MTNR1B P49286 1/20 0.40
PDE10A Q9Y233 3/20 0.36
CYP3A4 P08684 2/20 0.34
CYP2D6 P10635 2/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2E1 P05181 1/20 0.34
CYP2C8 P10632 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2B6 P20813 1/20 0.34
CYP2C19 P33261 1/20 0.34
MAPT P10636 3/20 0.33
KDM4E B2RXH2 3/20 0.33
GAA P10253 3/20 0.33
POLB P06746 2/20 0.33
PSMD14 O00487 1/20 0.33
ALDH1A1 P00352 3/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
DYRK1A Q13627 4/20 0.32
ADORA2A P29274 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15975203 0.95 PDE10A (0.38) MTNR1AMTNR1BPDE10ACYP3A4CYP2D6
SCHEMBL11979702 0.83 PDE10A (0.39) PDE10ACYP3A4CYP2D6CYP1A2CYP2E1
SCHEMBL11978295 0.82 PDE10A (0.37) PDE10ACYP3A4CYP2D6CYP1A2CYP2E1
SCHEMBL15975201 0.82 PDE10A (0.38) MTNR1AMTNR1BPDE10ACYP3A4CYP2D6
SCHEMBL11979697 0.81 TUBB4A (0.43) MTNR1AMTNR1BPDE10ACYP3A4CYP2D6
SCHEMBL15975133 0.80 PDE10A (0.37) PDE10AMAPTKDM4EALDH1A1DYRK1A
SCHEMBL15975129 0.79 MTNR1A (0.41) MTNR1AMTNR1BPDE10ACYP3A4CYP2D6
SCHEMBL11979709 0.79 CYP19A1 (0.48) PDE10A
SCHEMBL11979711 0.79 PDE10A (0.39) PDE10ACYP3A4CYP2D6CYP1A2MAPT
SCHEMBL4568577 0.78 MTNR1A (0.48) MTNR1AMTNR1BMAPTKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8815903-B2 Indole derivative and pharmacologically acceptable salt thereof KISSEI PHARMACEUTICAL CO., LTD. (JP) 2014-08-26 US disclosed
US-8815903-B2 Indole derivative and pharmacologically acceptable salt thereof KISSEI PHARMACEUTICAL CO., LTD. (JP) 2014-08-26 US disclosed