SCHEMBL15975815

SCHEMBL15975815

COc1cc(-c2nn3c(-c4cnc(N)c(C(C)(F)F)c4)c(C)nc3s2)ccc1OCC(=O)N(C)C

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 13/20 0.53
PIK3CD O00329 1/20 0.48
PIK3CB P42338 1/20 0.48
PIK3CG P48736 1/20 0.48
KDR P35968 3/20 0.37
KDM4E B2RXH2 2/20 0.35
TSHR P16473 2/20 0.35
MAPK1 P28482 2/20 0.35
USP2 O75604 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
HSD17B10 Q99714 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
DCTPP1 Q9H773 1/20 0.35
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL532165 0.95 PIK3CA (0.55) PIK3CAPIK3CDPIK3CBPIK3CGKDR
SCHEMBL15975808 0.89 PIK3CA (0.66) PIK3CAPIK3CDPIK3CBPIK3CGKDM4E
SCHEMBL2123270 0.84 PIK3CA (0.52) PIK3CAPIK3CDPIK3CBPIK3CGKDR
SCHEMBL532283 0.83 PIK3CA (0.67) PIK3CAPIK3CDPIK3CBPIK3CGKDM4E
SCHEMBL15975823 0.81 PIK3CA (0.52) PIK3CAPIK3CDPIK3CBPIK3CG
SCHEMBL532071 0.81 PIK3CA (0.55) PIK3CAPIK3CDPIK3CBPIK3CGKDM4E
SCHEMBL532397 0.79 PIK3CA (0.57) PIK3CAPIK3CDPIK3CBPIK3CG
SCHEMBL15976340 0.79 PIK3CA (0.51) PIK3CAPIK3CDPIK3CBPIK3CGLMNA
SCHEMBL2616035 0.79 PIK3CA (0.54) PIK3CAPIK3CDPIK3CBPIK3CGKDM4E
SCHEMBL533077 0.76 PIK3CA (0.53) PIK3CAPIK3CDPIK3CBPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8815918-B2 Imidazo [2, 1-B] [1, 3, 4] thiadiazole derivatives CENTRO NACIONAL DE INVESTIGACIONES ONCOLOGICAS (CNIO) (ES) 2014-08-26 US disclosed