SCHEMBL15975808

SCHEMBL15975808

COc1ccc(-c2nn3c(-c4cnc(N)c(C(C)(F)F)c4)c(C)nc3s2)cc1OC

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 12/20 0.66
PIK3CD O00329 1/20 0.59
PIK3CB P42338 1/20 0.59
PIK3CG P48736 1/20 0.59
KDM4E B2RXH2 5/20 0.44
ALDH1A1 P00352 5/20 0.44
MAPK1 P28482 4/20 0.44
TSHR P16473 2/20 0.44
LMNA P02545 2/20 0.44
HSD17B10 Q99714 2/20 0.44
USP2 O75604 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
DCTPP1 Q9H773 3/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
HPGD P15428 4/20 0.41
SIRT1 Q96EB6 1/20 0.41
KDM4C Q9H3R0 1/20 0.41
PKM P14618 1/20 0.40
STAT6 P42226 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL532283 0.94 PIK3CA (0.67) PIK3CAPIK3CDPIK3CBPIK3CGKDM4E
SCHEMBL15975815 0.89 PIK3CA (0.53) PIK3CAPIK3CDPIK3CBPIK3CGKDM4E
SCHEMBL15975823 0.86 PIK3CA (0.52) PIK3CAPIK3CDPIK3CBPIK3CG
SCHEMBL532397 0.86 PIK3CA (0.57) PIK3CAPIK3CDPIK3CBPIK3CG
SCHEMBL532475 0.83 PIK3CA (0.77) PIK3CAPIK3CDPIK3CBPIK3CGKDM4E
SCHEMBL532165 0.83 PIK3CA (0.55) PIK3CAPIK3CDPIK3CBPIK3CGKDM4E
SCHEMBL532071 0.82 PIK3CA (0.55) PIK3CAPIK3CDPIK3CBPIK3CGKDM4E
SCHEMBL15975822 0.81 PIK3CA (0.80) PIK3CAPIK3CDPIK3CBPIK3CGKDM4E
SCHEMBL15976340 0.81 PIK3CA (0.51) PIK3CAPIK3CDPIK3CBPIK3CGLMNA
SCHEMBL532676 0.81 PIK3CA (0.79) PIK3CAKDM4EALDH1A1MAPK1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8815918-B2 Imidazo [2, 1-B] [1, 3, 4] thiadiazole derivatives CENTRO NACIONAL DE INVESTIGACIONES ONCOLOGICAS (CNIO) (ES) 2014-08-26 US disclosed