SCHEMBL15975823

SCHEMBL15975823

COc1cc(-c2nn3c(-c4cnc(N)c(C(C)(F)F)c4)c(C)nc3s2)ccc1OCCN1CCOCC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 9/20 0.52
PIK3CD O00329 1/20 0.46
PIK3CB P42338 1/20 0.46
PIK3CG P48736 1/20 0.46
HTR2C P28335 2/20 0.42
HTR2B P41595 2/20 0.42
HTR2A P28223 1/20 0.42
KIT P10721 1/20 0.41
PRKAB2 O43741 1/20 0.40
PRKAG1 P54619 1/20 0.40
PRKAA2 P54646 1/20 0.40
PRKAA1 Q13131 1/20 0.40
PRKAG3 Q9UGI9 1/20 0.40
PRKAG2 Q9UGJ0 1/20 0.40
PRKAB1 Q9Y478 1/20 0.40
ADORA2A P29274 1/20 0.40
QPCT Q16769 1/20 0.39
QPCTL Q9NXS2 1/20 0.39
SCD O00767 1/20 0.39
MAP3K11 Q16584 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL533077 0.95 PIK3CA (0.53) PIK3CAPIK3CDPIK3CBPIK3CGHTR2C
SCHEMBL15975808 0.86 PIK3CA (0.66) PIK3CAPIK3CDPIK3CBPIK3CG
SCHEMBL533078 0.85 PIK3CA (0.46) PIK3CAPIK3CDPIK3CBPIK3CGHTR2C
SCHEMBL15975815 0.81 PIK3CA (0.53) PIK3CAPIK3CDPIK3CBPIK3CG
SCHEMBL532283 0.81 PIK3CA (0.67) PIK3CAPIK3CDPIK3CBPIK3CG
SCHEMBL532071 0.78 PIK3CA (0.55) PIK3CAPIK3CDPIK3CBPIK3CG
SCHEMBL15976340 0.77 PIK3CA (0.51) PIK3CAPIK3CDPIK3CBPIK3CG
SCHEMBL532165 0.76 PIK3CA (0.55) PIK3CAPIK3CDPIK3CBPIK3CG
SCHEMBL532397 0.76 PIK3CA (0.57) PIK3CAPIK3CDPIK3CBPIK3CG
SCHEMBL532475 0.72 PIK3CA (0.77) PIK3CAPIK3CDPIK3CBPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8815918-B2 Imidazo [2, 1-B] [1, 3, 4] thiadiazole derivatives CENTRO NACIONAL DE INVESTIGACIONES ONCOLOGICAS (CNIO) (ES) 2014-08-26 US disclosed