SCHEMBL16004121

SCHEMBL16004121

CCN(Cc1ccc2c(c1)CN(C(=O)c1ccccc1O)CCO2)C(C)=O

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 4/20 0.40
PIK3CA P42336 7/20 0.39
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
HSP90AA1 P07900 2/20 0.36
HSP90AB1 P08238 2/20 0.36
POLB P06746 1/20 0.36
CHRM5 P08912 1/20 0.36
CREBBP Q92793 1/20 0.36
BCL2 P10415 1/20 0.35
BAD Q92934 1/20 0.35
GPR142 Q7Z601 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16004118 0.83 PIK3CA (0.47) RIPK1PIK3CAGPR142
SCHEMBL16004128 0.81 PIK3CA (0.49) RIPK1PIK3CACREBBP
SCHEMBL16004291 0.80 MAPT (0.47) RIPK1NPC1RAB9APOLBCREBBP
SCHEMBL16004069 0.80 GPR142 (0.59) RIPK1NPC1RAB9ACREBBPGPR142
SCHEMBL16004060 0.79 LMNA (0.43) RIPK1PIK3CANPC1BCL2GPR142
SCHEMBL16003965 0.77 CHRM5 (0.40) RIPK1POLBCHRM5
SCHEMBL16004307 0.77 PIK3CA (0.40) RIPK1PIK3CANPC1RAB9AHSP90AA1
SCHEMBL16004052 0.76 PIK3CA (0.52) RIPK1PIK3CA
SCHEMBL16004102 0.76 PIK3CA (0.41) RIPK1PIK3CANPC1RAB9AHSP90AA1
SCHEMBL16004082 0.75 MC4R (0.38) RIPK1POLBCHRM5GPR142

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014133414-A2 HETEROCYCLIC TGR5 BILE ACID RECEPTOR AGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR THE PRODUCTION AND USE THEREOF АЛЛА ХЕМ ЛЛС (US) 2014-09-04 WO disclosed