SCHEMBL16004128

SCHEMBL16004128

CCN(Cc1ccc2c(c1)CN(C(=O)c1cccnc1)CCO2)C(C)=O

nearest known ligand 0.49

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 9/20 0.49
TDP1 Q9NUW8 2/20 0.46
KDM4E B2RXH2 1/20 0.46
HPGD P15428 1/20 0.44
RIPK1 Q13546 2/20 0.41
CTNNB1 P35222 1/20 0.39
WNT3A P56704 1/20 0.39
AHR P35869 1/20 0.39
GAA P10253 1/20 0.39
CREBBP Q92793 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16004118 0.90 PIK3CA (0.47) PIK3CARIPK1
SCHEMBL16004232 0.86 PIK3CA (0.49) PIK3CATDP1KDM4EHPGDRIPK1
SCHEMBL16004415 0.85 GPR142 (0.51)
SCHEMBL16004121 0.81 RIPK1 (0.40) PIK3CARIPK1CREBBP
SCHEMBL16004055 0.79 PIK3CA (0.49) PIK3CARIPK1
SCHEMBL16004052 0.78 PIK3CA (0.52) PIK3CAHPGDRIPK1GAA
SCHEMBL16004291 0.76 MAPT (0.47) TDP1KDM4EHPGDRIPK1CREBBP
SCHEMBL16004282 0.75 GPR142 (0.54)
SCHEMBL16004069 0.74 GPR142 (0.59) RIPK1CREBBP
SCHEMBL16004054 0.73 PIK3CA (0.49) PIK3CAHPGDRIPK1CREBBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014133414-A2 HETEROCYCLIC TGR5 BILE ACID RECEPTOR AGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR THE PRODUCTION AND USE THEREOF АЛЛА ХЕМ ЛЛС (US) 2014-09-04 WO disclosed