SCHEMBL16004289

SCHEMBL16004289

CCN(Cc1ccc2c(c1)CN(C(=O)Nc1ccsc1C(=O)O)CCO2)C(=O)C(C)C

nearest known ligand 0.41

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ABCC1 P33527 1/20 0.41
GPR142 Q7Z601 13/20 0.39
RIPK1 Q13546 2/20 0.37
CREBBP Q92793 2/20 0.37
RYR2 Q92736 1/20 0.36
FAAH O00519 1/20 0.35
CYP2D6 P10635 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16004288 0.92 ALDH1A1 (0.44) GPR142RIPK1RYR2
SCHEMBL16004075 0.91 ABCC1 (0.43) ABCC1GPR142RIPK1CREBBPRYR2
SCHEMBL16004284 0.85 GPR142 (0.42) GPR142CREBBPRYR2FAAHCYP2D6
SCHEMBL16004287 0.83 KMT2A (0.46) GPR142RYR2
SCHEMBL16004276 0.81 CREBBP (0.40) GPR142RIPK1CREBBPRYR2FAAH
SCHEMBL16004279 0.76 ALDH1A1 (0.46) GPR142RYR2
SCHEMBL16003991 0.76 ALDH1A1 (0.47) GPR142RYR2
SCHEMBL16004421 0.76 GPR142 (0.43) GPR142
SCHEMBL16004069 0.75 GPR142 (0.59) GPR142RIPK1CREBBPFAAH
SCHEMBL16004066 0.74 TAAR1 (0.45) GPR142RIPK1CREBBPFAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014133414-A2 HETEROCYCLIC TGR5 BILE ACID RECEPTOR AGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR THE PRODUCTION AND USE THEREOF АЛЛА ХЕМ ЛЛС (US) 2014-09-04 WO disclosed