SCHEMBL16004332

SCHEMBL16004332

O=S(=O)(c1cccc2nsnc12)N1CCOc2ccc(COCc3ccc(F)cc3)cc2C1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 5/20 0.50
MAPK1 P28482 2/20 0.50
USP2 O75604 1/20 0.50
POLB P06746 1/20 0.50
KMT2A Q03164 4/20 0.45
ALDH1A1 P00352 4/20 0.45
LMNA P02545 3/20 0.45
MEN1 O00255 2/20 0.45
CYP1A2 P05177 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.44
TP53 P04637 1/20 0.42
HSD17B10 Q99714 1/20 0.41
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16004329 0.93 MAPK1 (0.54) SMN1; SMN2MAPK1USP2KMT2AALDH1A1
SCHEMBL16004257 0.80 PKM (0.50) MAPK1KMT2AALDH1A1LMNAMEN1
SCHEMBL16004327 0.80 PKM (0.51) SMN1; SMN2USP2POLBKMT2AALDH1A1
SCHEMBL16004019 0.78 PKM (0.44) SMN1; SMN2MAPK1POLBKMT2AALDH1A1
SCHEMBL16004012 0.78 NPC1 (0.41) MAPK1POLBKMT2AALDH1A1LMNA
SCHEMBL16004260 0.75 CCR3 (0.50) MAPK1USP2KMT2AALDH1A1LMNA
SCHEMBL16004333 0.74 PKM (0.47) SMN1; SMN2MAPK1ALDH1A1LMNAL3MBTL1
SCHEMBL16004330 0.73 PKM (0.46) SMN1; SMN2USP2KMT2AALDH1A1LMNA
SCHEMBL16004229 0.72 PKM (0.46) MAPK1KMT2AALDH1A1LMNACYP1A2
SCHEMBL16004107 0.72 PKM (0.45) SMN1; SMN2KMT2AALDH1A1LMNAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014133414-A2 HETEROCYCLIC TGR5 BILE ACID RECEPTOR AGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR THE PRODUCTION AND USE THEREOF АЛЛА ХЕМ ЛЛС (US) 2014-09-04 WO disclosed