SCHEMBL16004333

SCHEMBL16004333

O=S(=O)(c1cc(F)cc(F)c1)N1CCOc2ccc(COCc3cccc(F)c3)cc2C1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PKM P14618 8/20 0.47
PKLR P30613 5/20 0.47
MAPK1 P28482 1/20 0.43
ALDH1A1 P00352 1/20 0.41
GPR142 Q7Z601 1/20 0.40
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
RORC P51449 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.37
MAOB P27338 1/20 0.37
GRM5 P41594 1/20 0.37
NTRK1 P04629 1/20 0.37
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
LMNA P02545 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16004019 0.91 PKM (0.44) PKMPKLRMAPK1ALDH1A1SMN1; SMN2
SCHEMBL16004231 0.90 PKM (0.53) PKMPKLRALDH1A1SMN1; SMN2NPSR1
SCHEMBL16004017 0.90 PKM (0.44) PKMPKLRMAPK1ALDH1A1GPR142
SCHEMBL16004230 0.89 PKM (0.46) PKMPKLRMAPK1ALDH1A1GPR142
SCHEMBL16004336 0.87 PKM (0.52) PKMPKLRMAPK1ALDH1A1SMN1; SMN2
SCHEMBL16004331 0.87 PKM (0.47) PKMPKLRMAPK1ALDH1A1GPR142
SCHEMBL16004012 0.87 NPC1 (0.41) PKMPKLRMAPK1ALDH1A1GPR142
SCHEMBL16004015 0.86 RORC (0.42) PKMPKLRMAPK1ALDH1A1HTT
SCHEMBL16004327 0.85 PKM (0.51) PKMPKLRALDH1A1SMN1; SMN2RORC
SCHEMBL16004255 0.83 L3MBTL1 (0.44) PKMPKLRMAPK1GPR142SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014133414-A2 HETEROCYCLIC TGR5 BILE ACID RECEPTOR AGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR THE PRODUCTION AND USE THEREOF АЛЛА ХЕМ ЛЛС (US) 2014-09-04 WO disclosed