SCHEMBL16004257

SCHEMBL16004257

O=S(=O)(c1ccc(F)cc1F)N1CCOc2ccc(COCc3ccc(F)cc3)cc2C1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PKM P14618 7/20 0.50
PKLR P30613 4/20 0.50
CNR1 P21554 2/20 0.39
RIPK1 Q13546 1/20 0.39
NTRK1 P04629 3/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPT P10636 1/20 0.39
LMNA P02545 2/20 0.37
MEN1 O00255 1/20 0.37
MAPK1 P28482 1/20 0.37
KMT2A Q03164 1/20 0.37
RORC P51449 1/20 0.37
MAOB P27338 1/20 0.35
GRM5 P41594 1/20 0.35
KDM2B Q8NHM5 1/20 0.35
NR3C2 P08235 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16004326 0.88 PKM (0.46) PKMPKLRCNR1RIPK1NTRK1
SCHEMBL16004327 0.88 PKM (0.51) PKMPKLRNTRK1ALDH1A1LMNA
SCHEMBL16004019 0.86 PKM (0.44) PKMPKLRRIPK1NTRK1ALDH1A1
SCHEMBL16004012 0.85 NPC1 (0.41) PKMPKLRRIPK1NTRK1ALDH1A1
SCHEMBL16004260 0.82 CCR3 (0.50) ALDH1A1MAPTLMNAMEN1MAPK1
SCHEMBL16004338 0.81 LMNA (0.39) PKMPKLRCNR1RIPK1NTRK1
SCHEMBL16004332 0.80 SMN1; SMN2 (0.50) ALDH1A1MAPTLMNAMEN1MAPK1
SCHEMBL16004330 0.80 PKM (0.46) PKMPKLRALDH1A1LMNAMEN1
SCHEMBL16004229 0.79 PKM (0.46) PKMPKLRALDH1A1MAPTLMNA
SCHEMBL16004333 0.79 PKM (0.47) PKMPKLRNTRK1ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014133414-A2 HETEROCYCLIC TGR5 BILE ACID RECEPTOR AGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR THE PRODUCTION AND USE THEREOF АЛЛА ХЕМ ЛЛС (US) 2014-09-04 WO disclosed