SCHEMBL16004752

SCHEMBL16004752

NCc1cc(F)ccc1Oc1ccc2[nH]ncc2c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 2/20 0.43
CTNNB1 P35222 1/20 0.41
WNT3A P56704 1/20 0.41
TRPA1 O75762 3/20 0.41
MAOB P27338 2/20 0.40
RAB9A P51151 2/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
KDM4E B2RXH2 1/20 0.40
ROCK2 O75116 1/20 0.40
ALDH1A1 P00352 1/20 0.40
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.40
HPGD P15428 1/20 0.40
HIF1A Q16665 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
EPAS1 Q99814 1/20 0.40
HTR2A P28223 5/20 0.39
SLC6A4 P31645 5/20 0.39
KCNH2 Q12809 5/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5043115 0.83 ROCK1 (0.52) ROCK1CTNNB1WNT3ATRPA1RAB9A
SCHEMBL378733 0.78 AR (0.46) ROCK1TRPA1EPAS1KCNH2
SCHEMBL5407364 0.75 MEN1 (0.46) ROCK1CTNNB1WNT3ATRPA1MAOB
SCHEMBL2876364 0.75 ROCK1 (0.58) ROCK1TRPA1MAOBRAB9AMEN1
SCHEMBL28707122 0.74 NOS1 (0.46) ROCK1CTNNB1WNT3ATRPA1MAOB
SCHEMBL5413417 0.73 GAA (0.59) ROCK1TRPA1RAB9AMEN1KMT2A
SCHEMBL12328667 0.73 MAP4K4 (0.40) HTR2ASLC6A4KCNH2
SCHEMBL3497213 0.72 TRPA1 (0.59) ROCK1CTNNB1WNT3ATRPA1MAOB
SCHEMBL5417525 0.72 SLC6A4 (0.55) TRPA1MEN1KMT2AHTR2ASLC6A4
Hydrochloric Acid SCHEMBL2450168 0.72 MAP4K4 (0.40) HTR2ASLC6A4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014134313-A1 INTERMEDIATES FOR USE IN THE PREPARATION OF INDAZOLE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF ARRAY BIOPHARMA INC. (US) 2014-09-04 WO disclosed