SCHEMBL16004998

SCHEMBL16004998

CCCCOc1c(Cl)cc(F)cc1C=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ORAI1 Q96D31 1/20 0.40
THRA P10827 3/20 0.39
THRB P10828 3/20 0.39
HTT P42858 1/20 0.38
RECQL P46063 1/20 0.38
ESR1 P03372 1/20 0.37
S1PR2 O95136 1/20 0.36
S1PR1 P21453 1/20 0.36
S1PR3 Q99500 1/20 0.36
LPAR2 Q9HBW0 1/20 0.36
CCNB2 O95067 2/20 0.36
CCNE2 O96020 2/20 0.36
CDK1 P06493 2/20 0.36
CDK4 P11802 2/20 0.36
CCNB1 P14635 2/20 0.36
CCND1 P24385 2/20 0.36
CCNE1 P24864 2/20 0.36
CDK2 P24941 2/20 0.36
CCND2 P30279 2/20 0.36
CCND3 P30281 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16005185 0.84 ORAI1 (0.54) ORAI1THRATHRBRECQLS1PR2
SCHEMBL16005078 0.82 THRA (0.42) ORAI1THRATHRBS1PR2S1PR1
SCHEMBL16005293 0.81 ORAI1 (0.38) ORAI1THRATHRBS1PR2S1PR1
SCHEMBL16005448 0.79 ORAI1 (0.52) ORAI1THRATHRBRECQLS1PR2
SCHEMBL30310598 0.77 ERN1 (0.40) KMT2AALDH1A1L3MBTL1TDP1ERN1
SCHEMBL1748304 0.77 ERN1 (0.40) KMT2AALDH1A1L3MBTL1TDP1ERN1
SCHEMBL17513175 0.76 ORAI1 (0.56) ORAI1HTTRECQLKMT2AALDH1A1
SCHEMBL12243717 0.74 GAA (0.38) ORAI1HTTRECQLS1PR2S1PR1
SCHEMBL7290764 0.74 SRC (0.47) THRATHRBALDH1A1L3MBTL1TDP1
SCHEMBL18181889 0.73 ALDH1A1 (0.51) HTTALDH1A1L3MBTL1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2774914-B1 N-BENZYLANILINE DERIVATIVE AND USES THEREOF UNIV NANJING MEDICAL (CN) 2017-12-06 EP disclosed
US-9481636-B2 N-benzylaniline derivative and uses thereof NANJING MEDICAL UNIVERSITY (CN) 2016-11-01 US disclosed
US-20140303248-A1 N-BENZYLANILINE DERIVATIVE AND USES THEREOF Neurodawn Pharmaceutical Co., Ltd. (CN) 2014-10-09 US disclosed
EP-2774914-A1 N-BENZYLANILINE DERIVATIVE AND USES THEREOF Nanjing Medical University (CN) 2014-09-10 EP disclosed
CN-103086908-A N-benzylaniline derivatives and application thereof UNIV NANJING MEDICAL 2013-05-08 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140303248-A1 N-BENZYLANILINE DERIVATIVE AND USES THEREOF NLN, INA, TRPV1 ORAI1 169/4885THRA 4105/4885THRB 3829/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.