SCHEMBL1600943

SCHEMBL1600943

CC(C)[Si](OCc1cc(C(F)(F)F)ccc1C1(O)CCCCCC1)(C(C)C)C(C)C

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
SLC6A2 P23975 6/20 0.38
SLC6A4 P31645 6/20 0.38
SLC6A3 Q01959 5/20 0.34
CETP P11597 1/20 0.32
IDO1 P14902 1/20 0.32
FFAR4 Q5NUL3 1/20 0.31
CYP11B1 P15538 1/20 0.31
CYP11B2 P19099 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1600954 0.85 SLC6A4 (0.34) MEN1KMT2ASLC6A2SLC6A4SLC6A3
SCHEMBL1600421 0.84 MEN1 (0.40) MEN1KMT2ASLC6A2SLC6A4SLC6A3
SCHEMBL1600326 0.73 IDO1 (0.38) SLC6A2SLC6A4IDO1
SCHEMBL3958892 0.70 POLB (0.38) IDO1
SCHEMBL3952559 0.70 AR (0.39) SLC6A2SLC6A4IDO1CYP11B1CYP11B2
SCHEMBL1601333 0.69 TACR1 (0.35) MEN1KMT2AFFAR4
SCHEMBL1600514 0.69 IDO1 (0.33) MEN1KMT2ASLC6A2SLC6A4SLC6A3
SCHEMBL3411309 0.69 MEN1 (0.47) MEN1KMT2ASLC6A2SLC6A4SLC6A3
SCHEMBL3952842 0.68 TACR1 (0.33)
SCHEMBL3953613 0.68 PDE2A (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7919506-B2 Dibenzyl amine compounds and derivatives PFIZER INC. (US) 2011-04-05 US disclosed
US-7919506-B2 Dibenzyl amine compounds and derivatives PFIZER INC. (US) 2011-04-05 US disclosed
EP-1996564-A1 DIBENZYL AMINE COMPOUNDS AND DERIVATIVES Pfizer Products Incorporated (US) 2008-12-03 EP disclosed
WO-2007105050-A1 DIBENZYL AMINE COMPOUNDS AND DERIVATIVES PFIZER PRODUCTS INC. (US) 2007-09-20 WO disclosed
US-20070213371-A1 Dibenzyl Amine Compounds and Derivatives PFIZER INC 2007-09-13 US disclosed
US-20070213371-A1 Dibenzyl Amine Compounds and Derivatives PFIZER INC 2007-09-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070213371-A1 Dibenzyl Amine Compounds and Derivatives APOB, LDLR, CETP MEN1 1597/4885KMT2A 798/4885SLC6A2 949/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.