SCHEMBL16016196

SCHEMBL16016196

CNc1cccc(-c2ccc(S(=O)(=O)NC)cc2)n1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 6/20 0.52
SMN1; SMN2 Q16637 2/20 0.44
GAA P10253 1/20 0.44
CA12 O43570 2/20 0.43
CA1 P00915 2/20 0.43
CA2 P00918 2/20 0.43
CA3 P07451 2/20 0.43
CA4 P22748 2/20 0.43
CA6 P23280 2/20 0.43
CA5A P35218 2/20 0.43
CA7 P43166 2/20 0.43
CA9 Q16790 2/20 0.43
CA13 Q8N1Q1 2/20 0.43
CA14 Q9ULX7 2/20 0.43
CA5B Q9Y2D0 2/20 0.43
SCN9A Q15858 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.42
LMNA P02545 1/20 0.42
HTT P42858 1/20 0.42
ATR Q13535 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12188971 0.85 HSD11B1 (0.42) HSD11B1SMN1; SMN2GAACA12CA1
SCHEMBL2035381 0.84 ATR (0.48) HSD11B1SMN1; SMN2GAAATRATRIP
SCHEMBL12170349 0.81 ASIC3 (0.51) HSD11B1SMN1; SMN2GAACA12CA1
Hydrochloric Acid SCHEMBL1721752 0.80 ASIC3 (0.50) HSD11B1SMN1; SMN2GAACA12CA1
SCHEMBL29574989 0.78 SCN9A (0.47) SCN9AATRATRIPALDH1A1NR3C2
SCHEMBL1721714 0.78 SCN9A (0.47) SCN9AATRATRIPALDH1A1NR3C2
SCHEMBL5914189 0.76 MEN1 (0.60) CNR1
SCHEMBL12169973 0.75 ALDH1A1 (0.47) HSD11B1SMN1; SMN2GAALMNAHTT
Hydrochloric Acid SCHEMBL29100611 0.74 MEN1 (0.58) CNR1
SCHEMBL12169703 0.73 ALDH1A1 (0.52) SMN1; SMN2GAAL3MBTL1LMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3208272-A1 HETEROCYCLIC MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS Vertex Pharmaceuticals Incorporated (US) 2017-08-23 EP disclosed
EP-2774925-A1 Pharmaceutical composition containing a heterocyclic modulator of ATP-binding cassette transporters Vertex Pharmaceuticals Incorporated (US) 2014-09-10 EP disclosed