SCHEMBL16029367

SCHEMBL16029367

O=Cc1ccc(-c2cccc(Cl)c2Cl)o1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 2/20 0.57
SIRT1 Q96EB6 2/20 0.57
SIRT5 Q9NXA8 2/20 0.57
KDM4E B2RXH2 8/20 0.56
LMNA P02545 6/20 0.56
KMT2A Q03164 5/20 0.56
HPGD P15428 5/20 0.56
TP53 P04637 1/20 0.56
IGF1R P08069 1/20 0.56
ALDH1A1 P00352 10/20 0.53
MAPT P10636 7/20 0.53
MEN1 O00255 4/20 0.53
ALOX12 P18054 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
POLB P06746 6/20 0.51
L3MBTL1 Q9Y468 4/20 0.50
SMN1; SMN2 Q16637 3/20 0.50
TDP1 Q9NUW8 2/20 0.48
PPARG P37231 1/20 0.48
NCOA2 Q15596 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30861665 1.00 SIRT2 (0.57) SIRT2SIRT1SIRT5KDM4ELMNA
SCHEMBL1616299 0.86 KDM4E (0.58) KDM4ELMNAKMT2AHPGDIGF1R
SCHEMBL6420665 0.80 KDM4E (0.46) SIRT2SIRT1SIRT5KDM4ELMNA
SCHEMBL31358694 0.79 SIRT2 (0.67) SIRT2SIRT1SIRT5KDM4ELMNA
SCHEMBL6573721 0.75 SIRT2 (0.81) SIRT2SIRT1SIRT5KDM4ELMNA
SCHEMBL6009639 0.73 ALDH1A1 (0.47) SIRT2SIRT1SIRT5KDM4ELMNA
SCHEMBL31358825 0.72 HPGD (0.60) SIRT2SIRT1SIRT5KDM4ELMNA
SCHEMBL31358679 0.72 IGF1R (0.64) SIRT2SIRT1SIRT5KDM4ELMNA
SCHEMBL1728691 0.72 MAPT (0.64) KDM4ELMNAKMT2AHPGDIGF1R
SCHEMBL4697667 0.72 HPGD (0.65) KDM4ELMNAKMT2AHPGDTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115611868-A Furanamide derivative and preparation method and application thereof 山东大学 2023-01-17 CN claimed
WO-2024103400-A1 POLYCYCLIC COMPOUND AS GPR75 ACTIVATOR, PHARMACEUTICAL COMPOSITION COMPRISING SAME, AND USE THEREOF 水木未来(北京)科技有限公司 2024-05-23 WO disclosed
CN-117820303-A Tetrahydroacridine-9 carboxylic acid derivative and preparation method and application thereof 中国药科大学 2024-04-05 CN disclosed
CN-115611868-A Furanamide derivative and preparation method and application thereof 山东大学 2023-01-17 CN disclosed
EP-3226858-B1 IMIDAZOLE-BASED ANTIMICROBIAL AGENTS PROCOMCURE BIOTECH GMBH (AT) 2021-02-03 EP disclosed
US-10456379-B2 Imidazole-based antimicrobial agents PROCOMCURE BIOTECH GMBH (AT) 2019-10-29 US disclosed
US-10322110-B2 Imidazole-based antimicrobial agents PROCOMCURE BIOTECH GMBH (AT) 2019-06-18 US disclosed
US-10011578-B2 Compounds for stabilizing ryanodine receptors from aberrant levels of calcium release ROSALIND FRANKLIN UNIVERSITY OF MEDICINE AND SCIENCE (US) 2018-07-03 US disclosed
US-20180022722-A1 Compounds for Stabilizing Ryanodine Receptors from Aberrant Levels of Calcium Release ROSALIND FRANKLIN UNIVERSITY OF MEDICINE AND SCIENCE 2018-01-25 US disclosed
US-20170368032-A1 Imidazole-Based Antimicrobial Agents PROCOMCURE BIOTECH GMBH (AT) 2017-12-28 US disclosed
US-20170334887-A1 Imidazole-Based Antimicrobial Agents PROCOMCURE BIOTECH GMBH (AT) 2017-11-23 US disclosed
EP-3226858-A1 IMIDAZOLE-BASED ANTIMICROBIAL AGENTS Procomcure Biotech GmbH (AT) 2017-10-11 EP disclosed
US-9725429-B2 Furanyl-imine and thiofuranyl-imine compounds for stabilizing ryanodine receptors from aberrant levels of calcium release ROSALIND FRANKLIN UNIVERSITY OF MEDICINE AND SCIENCE (US) 2017-08-08 US disclosed
WO-2016087616-A1 IMIDAZOLE-BASED ANTIMICROBIAL AGENTS PROCOMCURE BIOTECH GMBH (AT) 2016-06-09 WO disclosed
WO-2016087618-A1 IMIDAZOLE-BASED ANTIMICROBIAL AGENTS PROCOMCURE BIOTECH GMBH (AT) 2016-06-09 WO disclosed
US-20160024038-A1 Compounds For Stabilizing Ryanodine Receptors From Aberrant Levels Of Calcium Release ROSALIND FRANKLIN UNIVERSITY OF MEDICINE AND SCIENCE 2016-01-28 US disclosed
EP-2968229-A1 COMPOUNDS FOR STABILIZING RYANODINE RECEPTORS FROM ABERRANT LEVELS OF CALCIUM RELEASE Rosalind Franklin University of Medicine and Science (US) 2016-01-20 EP disclosed
US-9102645-B2 Compounds for stabilizing ryanodine receptors from aberrant levels of calcium release ROSALIND FRANKLIN UNIVERSITY OF MEDICINE AND SCIENCE (US) 2015-08-11 US disclosed
WO-2014144654-A1 COMPOUNDS FOR STABILIZING RYANODINE RECEPTORS FROM ABERRANT LEVELS OF CALCIUM RELEASE ROSALIND FRANKLIN UNIVERSITY OF MEDICINE AND SCIENCE (US) 2014-09-18 WO disclosed
US-20140275112-A1 Compounds For Stabilizing Ryanodine Receptors From Aberrant Levels Of Calcium Release ROSALIND FRANKLIN UNIVERSITY OF MEDICINE AND SCIENCE (US) 2014-09-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180022722-A1 Compounds for Stabilizing Ryanodine Receptors from Aberrant Levels of Calcium Release CHERP, RYR1, RYR2 SIRT2 1409/4885SIRT1 555/4885SIRT5 2283/4885
US-20170334887-A1 Imidazole-Based Antimicrobial Agents TLR5, NISCH, SLC11A2 SIRT2 1043/4885SIRT1 802/4885SIRT5 156/4885
US-20140275112-A1 Compounds For Stabilizing Ryanodine Receptors From Aberrant Levels Of Calcium Release CHERP, RYR1, RYR2 SIRT2 1409/4885SIRT1 555/4885SIRT5 2283/4885
US-10456379-B2 Imidazole-based antimicrobial agents TLR5, NISCH, SLC11A2 SIRT2 1043/4885SIRT1 802/4885SIRT5 156/4885
US-10322110-B2 Imidazole-based antimicrobial agents ARG1, SLC11A2, IKZF3 SIRT2 1171/4885SIRT1 1602/4885SIRT5 486/4885
US-10011578-B2 Compounds for stabilizing ryanodine receptors from aberrant levels of calcium release CHERP, RYR1, RYR2 SIRT2 1409/4885SIRT1 555/4885SIRT5 2283/4885
US-20170368032-A1 Imidazole-Based Antimicrobial Agents TLR5, NISCH, SLC11A2 SIRT2 1043/4885SIRT1 802/4885SIRT5 156/4885
US-20160024038-A1 Compounds For Stabilizing Ryanodine Receptors From Aberrant Levels Of Calcium Release CHERP, RYR1, RYR2 SIRT2 1409/4885SIRT1 555/4885SIRT5 2283/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.