SCHEMBL16070101

SCHEMBL16070101

O=C(I)Cc1ccc(Br)cc1F

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 1/20 0.46
PDPK1 O15530 1/20 0.44
AKR1B1 P15121 8/20 0.42
P2RX7 Q99572 2/20 0.42
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41
HSD17B10 Q99714 1/20 0.41
PYCR1 P32322 1/20 0.41
AKR1A1 P14550 1/20 0.40
NPC1 O15118 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL538344 0.85 DGAT1 (0.55) DGAT1PDPK1AKR1B1P2RX7MEN1
SCHEMBL29574602 0.85 DGAT1 (0.46) DGAT1PDPK1AKR1B1P2RX7MEN1
SCHEMBL31551664 0.85 DGAT1 (0.55) DGAT1PDPK1AKR1B1P2RX7MEN1
SCHEMBL8696600 0.85 DGAT1 (0.46) DGAT1PDPK1AKR1B1P2RX7MEN1
SCHEMBL29574729 0.83 AKR1B1 (0.52) DGAT1PDPK1AKR1B1P2RX7MEN1
SCHEMBL5835 0.83 AKR1B1 (0.52) DGAT1PDPK1AKR1B1P2RX7MEN1
SCHEMBL8444 0.81 DGAT1 (0.46) DGAT1PDPK1AKR1B1P2RX7MEN1
SCHEMBL16257133 0.81 IDO1 (0.46) P2RX7
SCHEMBL12501525 0.79 DGAT1 (0.43) DGAT1PDPK1AKR1B1P2RX7MEN1
SCHEMBL22235337 0.79 DGAT1 (0.43) DGAT1PDPK1AKR1B1P2RX7MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014141187-A1 PYRIDINE DERIVATIVES AS REARRANGED DURING TRANSFECTION (RET) KINASE INHIBITORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2014-09-18 WO disclosed