SCHEMBL16070271

SCHEMBL16070271

COC(=O)c1cccc(C)c1N=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 1/20 0.47
TSHR P16473 2/20 0.47
LMNA P02545 1/20 0.47
ALDH1A1 P00352 2/20 0.46
HSD17B10 Q99714 2/20 0.46
CFTR P13569 1/20 0.46
KDM4E B2RXH2 4/20 0.44
POLB P06746 3/20 0.44
ATM Q13315 1/20 0.44
MYC P01106 1/20 0.44
MAPT P10636 5/20 0.43
KMT2A Q03164 3/20 0.43
MEN1 O00255 1/20 0.43
HTT P42858 1/20 0.43
MAPK10 P53779 1/20 0.43
PTK2B Q14289 1/20 0.43
NCOA1 Q15788 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
NCOA3 Q9Y6Q9 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8105878 0.81 NR4A2 (0.44) NR4A2TSHRLMNAALDH1A1HSD17B10
SCHEMBL10362667 0.81 NR4A2 (0.44) NR4A2TSHRLMNAALDH1A1HSD17B10
SCHEMBL10067848 0.79 ALDH1A1 (0.57) TSHRLMNAALDH1A1HSD17B10KDM4E
SCHEMBL10067845 0.78 ALDH1A1 (0.49) TSHRLMNAALDH1A1HSD17B10KDM4E
SCHEMBL524457 0.77 LMNA (0.53) NR4A2TSHRLMNAALDH1A1HSD17B10
SCHEMBL29047133 0.77 CYP1A2 (0.49) LMNAPOLBMAPTKMT2AMEN1
SCHEMBL29702037 0.77 TSHR (0.63) NR4A2TSHRLMNAALDH1A1HSD17B10
Dimethyl Phthalate SCHEMBL28079217 0.77 TSHR (0.63) NR4A2TSHRLMNAALDH1A1HSD17B10
SCHEMBL101601 0.77 TSHR (0.63) NR4A2TSHRLMNAALDH1A1HSD17B10
SCHEMBL16599381 0.76 POLB (0.55) NR4A2TSHRLMNAALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014143960-A1 TETRAHYDROISOQUINOLIN-2-YL-(QUINAZOLIN-4-YL) METHANONE COMPOUNDS AS CANCER CELL GROWTH INHIBITORS REXAHN PHARMACEUTICALS, INC. (US) 2014-09-18 WO disclosed