SCHEMBL16085545

SCHEMBL16085545

O=C(Nc1ccc(CN2CCOCC2)cc1)c1ccc(CN2CCc3ccccc3C2)cc1

nearest known ligand 0.79

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.79
KDM4E B2RXH2 1/20 0.79
NOD1 Q9Y239 13/20 0.79
TNF P01375 11/20 0.79
MEN1 O00255 6/20 0.79
KMT2A Q03164 6/20 0.79
RAB9A P51151 6/20 0.79
S1PR2 O95136 1/20 0.79
CYP2D6 P10635 1/20 0.79
MAPT P10636 1/20 0.79
CYP2C9 P11712 1/20 0.79
CYP2C19 P33261 1/20 0.79
HTT P42858 1/20 0.79
NOD2 Q9HC29 9/20 0.78
LMNA P02545 2/20 0.77
HIF1A Q16665 2/20 0.73
EPAS1 Q99814 2/20 0.73
NPC1 O15118 5/20 0.72
HPGD P15428 1/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16085384 0.93 NOD1 (0.75) SMN1; SMN2KDM4ENOD1TNFMEN1
SCHEMBL16085389 0.92 NOD1 (0.73) SMN1; SMN2KDM4ENOD1TNFMEN1
SCHEMBL16263700 0.90 SMN1; SMN2 (0.89) SMN1; SMN2KDM4ENOD1TNFMEN1
SCHEMBL16085655 0.89 NOD1 (0.73) SMN1; SMN2KDM4ENOD1TNFMEN1
SCHEMBL16085403 0.89 SMN1; SMN2 (1.00) SMN1; SMN2KDM4ENOD1TNFMEN1
SCHEMBL16060510 0.88 NOD1 (1.00) SMN1; SMN2KDM4ENOD1TNFMEN1
SCHEMBL21657710 0.85 HIF1A (1.00) SMN1; SMN2MEN1KMT2ARAB9AMAPT
SCHEMBL16062262 0.85 NOD1 (0.80) SMN1; SMN2KDM4ENOD1TNFMEN1
SCHEMBL16085532 0.83 NOD1 (0.72) SMN1; SMN2KDM4ENOD1TNFMEN1
SCHEMBL8769811 0.82 RAB9A (0.83) SMN1; SMN2MEN1KMT2ARAB9ACYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014145642-A9 NRF2 SMALL MOLECULE INHIBITORS FOR CANCER THERAPY THE JOHNS HOPKINS UNIVERSITY (US) 2014-11-13 WO disclosed
WO-2014145642-A2 NRF2 SMALL MOLECULE INHIBITORS FOR CANCER THERAPY THE JOHNS HOPKINS UNIVERSITY (US) 2014-09-18 WO disclosed
US-8728631-B2 Dendrimer compound and organic luminescent device employing the same SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2014-05-20 US disclosed