SCHEMBL16093387

SCHEMBL16093387

C/C=C/c1ccc(COc2ccc(F)cn2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CXCR2 P25025 1/20 0.43
ALDH1A1 P00352 2/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
GSK3B P49841 1/20 0.39
BACE1 P56817 1/20 0.39
LMNA P02545 2/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
ELOVL1 Q9BW60 1/20 0.37
GRM5 P41594 3/20 0.37
GABRA5 P31644 2/20 0.37
TSHR P16473 2/20 0.36
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
CTSL P07711 1/20 0.36
CTSB P07858 1/20 0.36
MAPT P10636 2/20 0.36
APP P05067 2/20 0.36
MAPK1 P28482 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15177157 0.93 L3MBTL1 (0.43) CXCR2ALDH1A1L3MBTL1GSK3BBACE1
SCHEMBL15177139 0.84 KDM4E (0.40) ALDH1A1LMNANPC1RAB9ASMN1; SMN2
SCHEMBL510483 0.82 ALDH1A1 (0.55) CXCR2ALDH1A1L3MBTL1GSK3BBACE1
SCHEMBL16093377 0.80 CXCR2 (0.45) CXCR2ALDH1A1LMNAELOVL1GRM5
SCHEMBL15177143 0.80 AKT1 (0.48) CXCR2L3MBTL1GSK3BBACE1NPC1
SCHEMBL1106865 0.80 TLR4 (0.56) CXCR2MAOB
SCHEMBL510296 0.80 TLR4 (0.56) CXCR2MAOB
SCHEMBL16093390 0.78 GRM5 (0.38) ALDH1A1L3MBTL1GSK3BBACE1LMNA
SCHEMBL510015 0.77 ALDH1A1 (0.65) CXCR2ALDH1A1L3MBTL1GSK3BBACE1
SCHEMBL28791339 0.76 CXCR2 (0.63) CXCR2ALDH1A1L3MBTL1GRM5GABRA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8841327-B2 Heterocycles substituted pyridine derivatives and antifungal agent containing thereof EISAI R&D MANAGEMENT CO., LTD. (JP) 2014-09-23 US disclosed