SCHEMBL16098699

SCHEMBL16098699

Cc1cc(O)cc2c1c1ccncc1n2CCN(C)C

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 2/20 0.44
ADORA2A P29274 1/20 0.44
CYP2D6 P10635 1/20 0.41
WEE1 P30291 5/20 0.37
HTR2A P28223 2/20 0.36
HTR2C P28335 2/20 0.36
DYRK1A Q13627 2/20 0.36
CHEK1 O14757 3/20 0.36
SRC P12931 1/20 0.36
KDM5A P29375 1/20 0.36
HASPIN Q8TF76 1/20 0.35
ROCK2 O75116 1/20 0.33
HTR1D P28221 1/20 0.33
CMA1 P23946 1/20 0.32
TDP2 O95551 2/20 0.32
TDP1 Q9NUW8 2/20 0.32
RPS6KA5 O75582 1/20 0.32
TERT O14746 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16100006 0.84 ADORA3 (0.41) ADORA3ADORA2ACYP2D6KDM5AHASPIN
SCHEMBL16097995 0.84 CYP2D6 (0.38) ADORA3ADORA2ACYP2D6WEE1HTR2A
SCHEMBL16099514 0.83 DYRK1A (0.49) ADORA3ADORA2ACYP2D6HTR2AHTR2C
SCHEMBL16099174 0.82 HASPIN (0.55) ADORA3ADORA2ACYP2D6KDM5AHASPIN
SCHEMBL16099273 0.81 ADORA3 (0.40) ADORA3ADORA2ADYRK1AKDM5AROCK2
SCHEMBL16099658 0.79 NFATC1 (0.43) ADORA3ADORA2AWEE1DYRK1ACHEK1
SCHEMBL16093943 0.77 NFATC1 (0.47) ADORA3ADORA2ACYP2D6WEE1DYRK1A
SCHEMBL8172390 0.73 CYP2D6 (0.70) CYP2D6TDP2TDP1TERT
SCHEMBL16099752 0.72 HASPIN (0.47) ADORA3ADORA2ACYP2D6HTR2AHTR2C
SCHEMBL16100067 0.71 ADORA3 (0.36) ADORA3ADORA2ADYRK1AKDM5ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2968284-A2 ALKYL-AMINE HARMINE DERIVATIVES FOR PROMOTING BONE GROWTH Osteoqc Inc. (CA) 2016-01-20 EP disclosed
WO-2014153203-A2 ALKYL-AMINE HARMINE DERIVATIVES FOR PROMOTING BONE GROWTH OSSIFI INC. (US) 2014-09-25 WO disclosed