SCHEMBL16097995

SCHEMBL16097995

CN(C)CCn1c2cnccc2c2c(C(F)(F)F)cc(O)cc21

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.38
ADORA3 P0DMS8 1/20 0.36
ADORA2A P29274 1/20 0.36
WEE1 P30291 4/20 0.35
CHEK1 O14757 3/20 0.34
SRC P12931 1/20 0.34
KDM5A P29375 1/20 0.33
HASPIN Q8TF76 1/20 0.33
HTR2A P28223 1/20 0.32
HTR2C P28335 1/20 0.32
DYRK1A Q13627 1/20 0.32
ROCK2 O75116 2/20 0.31
SCN9A Q15858 2/20 0.31
S1PR1 P21453 1/20 0.31
S1PR3 Q99500 1/20 0.31
CNR2 P34972 1/20 0.31
HTR1D P28221 1/20 0.31
TDP2 O95551 2/20 0.30
TDP1 Q9NUW8 2/20 0.30
GPBAR1 Q8TDU6 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16099365 0.85 CYP2D6 (0.35) CYP2D6ADORA3ADORA2AKDM5AHASPIN
SCHEMBL16099097 0.85 HASPIN (0.45) CYP2D6HASPINHTR2AHTR2CDYRK1A
SCHEMBL16098699 0.84 ADORA3 (0.44) CYP2D6ADORA3ADORA2AWEE1CHEK1
SCHEMBL2565027 0.82 HASPIN (0.49) CYP2D6ADORA3ADORA2AHASPINTDP1
SCHEMBL16099686 0.80 NFATC1 (0.41) CYP2D6WEE1CHEK1DYRK1ACNR2
SCHEMBL16097799 0.78 ADORA3 (0.33) ADORA3ADORA2AROCK2SCN9A
SCHEMBL16094165 0.77 HASPIN (0.41) CYP2D6HASPINHTR2AHTR2CDYRK1A
SCHEMBL16100179 0.74 PLK1 (0.43) CNR2
SCHEMBL16098616 0.72 ADORA3 (0.32) ADORA3ADORA2A
SCHEMBL16099514 0.70 DYRK1A (0.49) CYP2D6ADORA3ADORA2AHASPINHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2968284-A2 ALKYL-AMINE HARMINE DERIVATIVES FOR PROMOTING BONE GROWTH Osteoqc Inc. (CA) 2016-01-20 EP disclosed
WO-2014153203-A2 ALKYL-AMINE HARMINE DERIVATIVES FOR PROMOTING BONE GROWTH OSSIFI INC. (US) 2014-09-25 WO disclosed