SCHEMBL16100739

SCHEMBL16100739

CC(C)c1ccc(C(=O)C(C)(C)O)cc1.CCCCCCCCCCCCCCC(C)(C=O)Cc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
CTSK P43235 3/20 0.39
MBOAT4 Q96T53 1/20 0.37
MMP1 P03956 1/20 0.36
MMP9 P14780 1/20 0.36
MMP13 P45452 1/20 0.36
CTSL P07711 1/20 0.36
CTSB P07858 1/20 0.36
MLYCD O95822 1/20 0.35
CTSG P08311 2/20 0.35
CMA1 P23946 2/20 0.35
HTT P42858 2/20 0.35
LMNA P02545 1/20 0.35
PKM P14618 1/20 0.35
PRSS1 P07477 1/20 0.35
CTRB1 P17538 1/20 0.35
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6796742 0.80 CTSK (0.43) SMN1; SMN2CTSKMBOAT4MMP1MMP9
SCHEMBL4245984 0.80 CTSK (0.43) SMN1; SMN2CTSKMBOAT4MMP1MMP9
SCHEMBL28357907 0.79 CTSK (0.44) SMN1; SMN2CTSKMMP1MMP9MMP13
SCHEMBL16100740 0.76 RAB9A (0.41) NPC1RAB9ASMN1; SMN2MMP1MMP9
SCHEMBL5705633 0.76 THRA (0.50) MEN1KMT2A
SCHEMBL624141 0.75 CTSK (0.45) SMN1; SMN2CTSKMMP1MMP9MMP13
SCHEMBL1409972 0.74 CYP2C9 (0.49) NPC1RAB9ASMN1; SMN2MLYCDHTT
SCHEMBL8844556 0.71 RAB9A (0.42) NPC1RAB9ASMN1; SMN2HTTLMNA
Hexane SCHEMBL811498 0.71 CES1 (0.53) CTSGCMA1LMNAPRSS1CTRB1
SCHEMBL54909 0.71 CYP2C9 (0.50) RAB9ASMN1; SMN2HTTLMNAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2928895-B1 DERIVATIVES OF DIANHYDROHEXITOL AND THEIR USE AS CROSSLINKABLE COMPOSITIONS ROQUETTE FRERES (FR) 2020-01-08 EP disclosed
EP-3019501-B1 USE OF NOVEL COMPOUNDS DERIVED FROM 1,4:3,6 DIANHYDROHEXITOL FOR THE PRODUCTION OF POLYMER COATINGS ROQUETTE FRERES (FR) 2018-08-08 EP disclosed
EP-2928969-B1 CROSS-LINKABLE COMPOSITIONS BASED ON DIANHYDROHEXITOL COMPOUNDS ROQUETTE FRERES (FR) 2017-08-02 EP disclosed
EP-3019501-A1 USE OF NOVEL COMPOUNDS DERIVED FROM 1,4:3,6 DIANHYDROHEXITOL FOR THE PRODUCTION OF POLYMER COATINGS Roquette Frères (FR) 2016-05-18 EP disclosed
EP-2976399-A1 CROSS-LINKABLE COMPOSITIONS BASED ON COMPOUNDS OF (METH)ACRYLATED DERIVATIVES OF DIANHYDROHEXITOL Roquette Frères (FR) 2016-01-27 EP disclosed
WO-2015004381-A1 USE OF NOVEL COMPOUNDS DERIVED FROM 1,4:3,6 DIANHYDROHEXITOL FOR THE PRODUCTION OF POLYMER COATINGS ROQUETTE FRERES (FR) 2015-01-15 WO disclosed
WO-2014147340-A1 CROSS-LINKABLE COMPOSITIONS BASED ON COMPOUNDS OF (METH)ACRYLATED DERIVATIVES OF DIANHYDROHEXITOL ROQUETTE FRERES (FR) 2014-09-25 WO disclosed