SCHEMBL16111402

SCHEMBL16111402

O=C(OCc1ccccc1)c1ccnn1-c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 5/20 0.50
KMT2A Q03164 3/20 0.50
SLC6A2 P23975 1/20 0.50
SLC6A3 Q01959 1/20 0.50
MAPT P10636 2/20 0.49
KDM4E B2RXH2 1/20 0.49
MAOB P27338 1/20 0.49
ADORA2A P29274 1/20 0.49
TSHR P16473 3/20 0.49
L3MBTL1 Q9Y468 3/20 0.48
LMNA P02545 2/20 0.48
ALDH1A1 P00352 4/20 0.46
HPGD P15428 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
POLB P06746 1/20 0.46
CASP3 P42574 2/20 0.44
SENP8 Q96LD8 2/20 0.44
SENP7 Q9BQF6 2/20 0.44
SENP6 Q9GZR1 2/20 0.44
JMJD6 Q6NYC1 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9681622 0.84 ALDH1A1 (0.57) KMT2AMAPTKDM4EADORA2ALMNA
SCHEMBL20646162 0.81 GPR52 (0.52) TDP1KMT2ASLC6A2SLC6A3MAPT
SCHEMBL18394893 0.78 TP53 (0.50) TDP1KMT2AMAPTKDM4ETSHR
SCHEMBL856957 0.76 POLB (0.52) MAPTKDM4EL3MBTL1ALDH1A1POLB
SCHEMBL5399902 0.75 MAPT (0.50) TDP1KMT2ASLC6A2SLC6A3MAPT
SCHEMBL5963082 0.74 ALDH1A1 (0.47) KDM4ELMNAALDH1A1HPGDRAB9A
Hydrochloric Acid SCHEMBL11893514 0.74 POLB (0.50) MAPTKDM4EL3MBTL1ALDH1A1POLB
SCHEMBL31582366 0.73 TDP1 (0.43) TDP1KMT2ASLC6A2SLC6A3MAPT
SCHEMBL31582374 0.73 TDP1 (0.43) TDP1KMT2ASLC6A2SLC6A3MAPT
SCHEMBL10242690 0.73 MAPK1 (0.51) ALDH1A1POLBMAPK1GLS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014159214-A1 HISTONE DEACETYLASE INHIBITORS AND COMPOSITIONS AND METHODS OF USE THEREOF CHDI FOUNDATION, INC. (US) 2014-10-02 WO disclosed