SCHEMBL16112985

SCHEMBL16112985

Cc1cc(-c2cccnc2)cc2c(N3CCc4ccc(C(=O)N5CC[C@H](F)C5)cc4C3)ncnc12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.38
MEN1 O00255 1/20 0.38
LMNA P02545 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
ALOX15 P16050 1/20 0.38
MAPK1 P28482 1/20 0.38
KMT2A Q03164 1/20 0.38
CLK4 Q9HAZ1 1/20 0.38
DPP4 P27487 1/20 0.38
DPP7 Q9UHL4 1/20 0.38
GBA1 P04062 1/20 0.38
GAA P10253 1/20 0.37
MAPT P10636 1/20 0.37
GHSR Q92847 1/20 0.37
AURKA O14965 2/20 0.37
RPS6KB1 P23443 2/20 0.37
AURKB Q96GD4 1/20 0.37
ABL1 P00519 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16112610 1.00 ALDH1A1 (0.38) ALDH1A1MEN1LMNACYP1A2CYP3A4
SCHEMBL16142175 0.93 VNN1 (0.40) ALDH1A1MEN1LMNACYP1A2CYP3A4
SCHEMBL16112190 0.92 AURKA (0.39) ALDH1A1MEN1LMNACYP1A2CYP3A4
SCHEMBL16142217 0.91 MAP4K4 (0.43) ALDH1A1MEN1LMNACYP1A2CYP3A4
SCHEMBL16142215 0.89 HPGD (0.44) ALDH1A1MEN1LMNACYP1A2CYP3A4
SCHEMBL16112357 0.88 ALDH1A1 (0.47) ALDH1A1MEN1LMNACYP1A2CYP3A4
SCHEMBL16142214 0.87 LMNA (0.45) ALDH1A1MEN1LMNACYP1A2CYP3A4
SCHEMBL16113563 0.86 GBA1 (0.45) ALDH1A1MEN1LMNACYP1A2CYP3A4
SCHEMBL16112172 0.85 AURKA (0.46) ALDH1A1MEN1LMNACYP1A2CYP3A4
SCHEMBL16113283 0.84 SCN9A (0.44) ALDH1A1MEN1LMNACYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014160177-A2 QUINAZOLINE INHIBITORS OF PI3K EXELIXIS, INC. (US) 2014-10-02 WO claimed
WO-2014160177-A2 QUINAZOLINE INHIBITORS OF PI3K EXELIXIS, INC. (US) 2014-10-02 WO disclosed