SCHEMBL16129491

SCHEMBL16129491

FC(F)(F)c1cc(C(F)(F)F)c2[nH]cnc2c1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.46
S1PR1 P21453 1/20 0.36
CDK1 P06493 2/20 0.35
CACNA1H O95180 3/20 0.34
CACNA1B Q00975 1/20 0.34
CACNA1C Q13936 1/20 0.34
MAPT P10636 1/20 0.34
QPCT Q16769 1/20 0.33
CDC7 O00311 3/20 0.33
DBF4 Q9UBU7 3/20 0.33
BRAF P15056 1/20 0.33
CTSS P25774 1/20 0.33
CTSK P43235 1/20 0.33
HCAR1 Q9BXC0 1/20 0.33
MET P08581 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24533998 0.80 ULK1 (0.39) PARP1CDK1MAPTBRAF
SCHEMBL11565241 0.80 PARP1 (0.45) PARP1S1PR1MAPTCDC7DBF4
SCHEMBL22361949 0.80 PARP1 (0.45) PARP1S1PR1MAPTCDC7DBF4
SCHEMBL31436452 0.80 CDK1 (0.36) PARP1S1PR1CDK1MAPTCDC7
SCHEMBL2298425 0.80 PARP1 (0.45) PARP1S1PR1MAPTCDC7DBF4
SCHEMBL2431453 0.76 PARP1 (0.42) PARP1S1PR1MAPTQPCTCDC7
SCHEMBL13759404 0.76 PARP1 (0.42) PARP1S1PR1CACNA1HMAPTQPCT
SCHEMBL13759405 0.76 PARP1 (0.45) PARP1S1PR1CDK1MAPTQPCT
SCHEMBL30792066 0.76 KIF11 (0.34) PARP1CDK1CDC7DBF4
SCHEMBL15093877 0.75 PARP1 (0.44) PARP1S1PR1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014153001-A1 COMBINATION THERAPY FOR TREATING CANCER Epizyme, Inc. (US) 2014-09-25 WO disclosed