SCHEMBL16130385

SCHEMBL16130385

C=CCCOC(=O)[C@H](C)N

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.41
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38
TDP1 Q9NUW8 1/20 0.36
PSMB5 P28074 1/20 0.34
ALOX15 P16050 1/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 3/20 0.33
CYP3A4 P08684 3/20 0.33
LMNA P02545 2/20 0.33
USP2 O75604 2/20 0.33
MAPT P10636 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
RECQL P46063 1/20 0.33
GRIN2D O15399 1/20 0.33
GRIN3B O60391 1/20 0.33
GRIN1 Q05586 1/20 0.33
GRIN2A Q12879 1/20 0.33
GRIN2B Q13224 1/20 0.33
GRIN2C Q14957 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16130358 0.88 ALDH1A1 (0.39) TSHRTDP1ALDH1A1CYP3A4LMNA
SCHEMBL16130378 0.86 ALDH1A1 (0.42) TSHRALDH1A1CYP3A4LMNAUSP2
SCHEMBL24049939 0.84 TSHR (0.38) TSHRCA2CA9TDP1PSMB5
SCHEMBL9301011 0.83 TSHR (0.43) TSHRCA2CA9TDP1PSMB5
SCHEMBL28496420 0.80
SCHEMBL905193 0.80
SCHEMBL1110727 0.80
SCHEMBL13785332 0.79 CHRNB2 (0.41) TSHRALOX15ALDH1A1CYP3A4LMNA
SCHEMBL14456617 0.79 TSHR (0.41) TSHRCA2CA9TDP1PSMB5
SCHEMBL19309165 0.79 DPP4 (0.43) TSHRCA2CA9TDP1PSMB5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021093860-A1 SUBSTITUTED BIS-TRICYCLIC COMPOUND, AND PHARMACEUTICAL COMPOSITION AND USE THEREOF 南京知和医药科技有限公司 2021-05-20 WO disclosed
US-8846638-B2 Macrocyclic nucleoside phosphoramidate derivatives ENANTA PHARMACEUTICALS, INC. (US) 2014-09-30 US disclosed
US-8846638-B2 Macrocyclic nucleoside phosphoramidate derivatives ENANTA PHARMACEUTICALS, INC. (US) 2014-09-30 US disclosed