SCHEMBL16147803

SCHEMBL16147803

O=C(O)c1ccc(NC(=O)c2cccc(C(F)(F)F)c2O)c(Cl)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PYGL P06737 3/20 0.52
KDM4E B2RXH2 1/20 0.50
PDK1 Q15118 1/20 0.50
PDK2 Q15119 1/20 0.50
PDK3 Q15120 1/20 0.50
PDK4 Q16654 1/20 0.50
PPARG P37231 3/20 0.49
NR1H4 Q96RI1 3/20 0.49
PPARD Q03181 2/20 0.49
P2RX1 P51575 1/20 0.47
P2RX4 Q99571 1/20 0.47
P2RX7 Q99572 1/20 0.47
TMPRSS4 Q9NRS4 1/20 0.47
PPARA Q07869 1/20 0.47
KCNK3 O14649 1/20 0.45
KCNK9 Q9NPC2 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C19 P33261 1/20 0.45
RAB9A P51151 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7341170 0.89 PYGL (0.58) PYGLKDM4EPDK1PDK2PDK3
SCHEMBL8314728 0.80 PYGL (0.62) PYGLKDM4EPDK1PDK2PDK3
SCHEMBL8314210 0.78 PYGL (0.64) PYGLKDM4EPDK1PDK2PDK3
SCHEMBL16147800 0.77 TMPRSS4 (0.59) PYGLPDK1PDK2PDK3PDK4
SCHEMBL27532598 0.77 MEN1 (0.59) PDK1PDK2PDK3PDK4PPARG
SCHEMBL8316647 0.76 PYGL (0.54) PYGLKDM4EPDK1PDK2PDK3
SCHEMBL16147472 0.75 NR1H4 (0.52) PYGLKDM4EPDK1PDK2PDK3
SCHEMBL8313578 0.75 PYGL (0.56) PYGLKDM4EPDK1PDK2PDK3
SCHEMBL20601791 0.75 KCNK3 (0.55) KDM4EPPARGNR1H4KCNK3KCNK9
SCHEMBL31585855 0.75 KCNK3 (0.55) KDM4EPPARGNR1H4KCNK3KCNK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014165816-A1 COMPOUNDS USEFUL FOR THE TREATMENT OF METABOLIC DISORDERS AND SYNTHESIS OF THE SAME NORTH CAROLINA CENTRAL UNIVERSITY (US) 2014-10-09 WO disclosed