SCHEMBL8314728

SCHEMBL8314728

O=C(O)c1ccc(NC(=O)c2ccc(F)cc2C(F)(F)F)c(Cl)c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PYGL P06737 5/20 0.62
ALOX15 P16050 4/20 0.52
PDK1 Q15118 1/20 0.51
PDK2 Q15119 1/20 0.51
PDK3 Q15120 1/20 0.51
PDK4 Q16654 1/20 0.51
RAB9A P51151 2/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C19 P33261 1/20 0.46
KCNK2 O95069 1/20 0.46
TP53 P04637 1/20 0.46
MAPT P10636 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
KDM4E B2RXH2 1/20 0.45
PPARG P37231 2/20 0.45
PPARD Q03181 2/20 0.45
NR1H4 Q96RI1 2/20 0.45
PPARA Q07869 1/20 0.45
GRM4 Q14833 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22871422 0.88 MAPT (0.48) PYGLRAB9ACYP1A2CYP2C19KCNK2
SCHEMBL7341170 0.85 PYGL (0.58) PYGLPDK1PDK2PDK3PDK4
SCHEMBL8317775 0.83 LMNA (0.47) PYGLALOX15PDK1PDK2PDK3
SCHEMBL27284321 0.82 KDM4E (0.55) ALOX15RAB9ACYP1A2CYP2C19TP53
SCHEMBL16148162 0.81 PYGL (0.62) PYGLALOX15PDK1PDK2PDK3
SCHEMBL7340569 0.80 PYGL (0.61) PYGLALOX15PDK1PDK2PDK3
SCHEMBL16147803 0.80 PYGL (0.52) PYGLPDK1PDK2PDK3PDK4
SCHEMBL31586268 0.78 KCNK2 (0.50) PYGLRAB9ACYP1A2CYP2C19KCNK2
SCHEMBL22871312 0.78 KCNK2 (0.50) PYGLRAB9ACYP1A2CYP2C19KCNK2
SCHEMBL1160893 0.76 AURKA (0.48) ALOX15MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0636625-B1 Tricyclic diazepines vasopressin and oxytocin antagonists AMERICAN CYANAMID CO (US) 1999-01-27 EP disclosed