SCHEMBL16148658

SCHEMBL16148658

COc1cc(/C=C(\C#N)C(=O)O)cc(NC(C)=O)c1O

nearest known ligand 0.54

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
EGFR P00533 7/20 0.54
ERBB2 P04626 6/20 0.54
DNM1 Q05193 5/20 0.54
KMT2A Q03164 4/20 0.51
MEN1 O00255 3/20 0.50
MAPT P10636 2/20 0.50
ALDH1A1 P00352 1/20 0.50
PTP4A3 O75365 1/20 0.48
PTP4A2 Q12974 1/20 0.48
PTP4A1 Q93096 1/20 0.48
CYP1A2 P05177 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16148661 1.00 EGFR (0.54) EGFRERBB2DNM1KMT2AMEN1
SCHEMBL8749247 0.86 DNM1 (0.61) EGFRERBB2DNM1KMT2AMEN1
SCHEMBL5164387 0.86 DNM1 (0.61) EGFRERBB2DNM1KMT2AMEN1
SCHEMBL16160400 0.85 ALDH1A1 (0.62) EGFRERBB2DNM1KMT2AMEN1
SCHEMBL7820539 0.83 DNM1 (0.70) EGFRERBB2DNM1KMT2AMEN1
SCHEMBL7820542 0.83 DNM1 (0.70) EGFRERBB2DNM1KMT2AMEN1
SCHEMBL8646383 0.77 KDM4E (0.56) DNM1KMT2AMEN1MAPTALDH1A1
SCHEMBL11761701 0.77 KDM4E (0.56) DNM1KMT2AMEN1MAPTALDH1A1
SCHEMBL9559164 0.77 EGFR (0.56) EGFRERBB2DNM1KMT2AMEN1
SCHEMBL29813583 0.76 EGFR (0.73) EGFRDNM1KMT2AMEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014164667-A1 DENGUE AND WEST NILE VIRUS PROTEASE INHIBITORS GEORGETOWN UNIVERSITY (US) 2014-10-09 WO disclosed