SCHEMBL16155308

SCHEMBL16155308

Cc1ccc2ncc(Cl)cc2c1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.50
CYP1A2 P05177 4/20 0.47
LMNA P02545 1/20 0.43
NCK1 P16333 1/20 0.41
BACE1 P56817 1/20 0.41
PDE3B Q13370 1/20 0.41
PDE3A Q14432 1/20 0.41
CYP2A6 P11509 2/20 0.41
NQO2 P16083 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
PSMB5 P28074 1/20 0.40
KDM4E B2RXH2 1/20 0.39
MET P08581 1/20 0.38
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8268977 0.84 ALDH1A1 (0.50) ALDH1A1CYP1A2LMNANCK1BACE1
SCHEMBL434860 0.84 CYP1A2 (0.57) ALDH1A1CYP1A2LMNAMEN1KMT2A
SCHEMBL4572536 0.83 CYP1A2 (0.65) ALDH1A1CYP1A2NCK1BACE1PDE3B
SCHEMBL24261121 0.76 ALDH1A1 (0.50) ALDH1A1CYP1A2NCK1BACE1PDE3B
SCHEMBL2000504 0.76 MAP4K4 (0.54) ALDH1A1CYP1A2NCK1BACE1CYP2A6
SCHEMBL16289890 0.76 ALDH1A1 (0.50) ALDH1A1CYP1A2NCK1BACE1PDE3B
SCHEMBL5509853 0.76 ALDH1A1 (0.50) ALDH1A1CYP1A2NCK1BACE1PDE3B
SCHEMBL2002584 0.76 ALDH1A1 (0.50) ALDH1A1CYP1A2LMNANCK1BACE1
SCHEMBL16962242 0.76 ALDH1A1 (0.50) ALDH1A1CYP1A2NCK1BACE1PDE3B
SCHEMBL1359776 0.76 MAP4K4 (0.46) ALDH1A1PDE3BPDE3AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2988597-B1 MACROLIDES AND METHODS OF THEIR PREPARATION AND USE HARVARD COLLEGE (US) 2022-06-08 EP disclosed
US-20170305953-A1 14-MEMBERED KETOLIDES AND METHODS OF THEIR PREPARATION AND USE PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2017-10-26 US disclosed
WO-2016161176-A1 METHODS FOR TREATING VIRAL INFECTIONS THE CALIFORNIA INSTITUTE FOR BIOMEDICAL RESEARCH (US) 2016-10-06 WO disclosed
WO-2016154591-A1 MACROLIDES WITH MODIFIED DESOSAMINE SUGARS AND USES THEREOF PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2016-09-29 WO disclosed
WO-2016057798-A1 14-MEMBERED KETOLIDES AND METHODS OF THEIR PREPARATION AND USE PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2016-04-14 WO disclosed
WO-2014165792-A2 MACROLIDES AND METHODS OF THEIR PREPARATION AND USE PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2014-10-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170305953-A1 14-MEMBERED KETOLIDES AND METHODS OF THEIR PREPARATION AND USE CYP51A1, HSD17B7, CYP11B1 ALDH1A1 1733/4885CYP1A2 117/4885LMNA 1699/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.