SCHEMBL16166247

SCHEMBL16166247

O=C1C[C@]2(C(=O)Nc3ccc(Cl)cc32)c2cnn(Cc3ccc(Cl)cc3)c2N1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 1/20 0.40
IDO1 P14902 2/20 0.36
CBX7 O95931 1/20 0.35
CDYL2 Q8N8U2 1/20 0.35
CDYL Q9Y232 1/20 0.35
CDY1; CDY1B Q9Y6F8 1/20 0.35
ALDH1A1 P00352 1/20 0.34
POLB P06746 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
HTR7 P34969 2/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.34
TSHR P16473 1/20 0.33
HTR2C P28335 1/20 0.33
HTR2B P41595 1/20 0.33
MGAM O43451 1/20 0.33
HTR1A P08908 1/20 0.33
GAA P10253 1/20 0.33
SI P14410 1/20 0.33
HTR2A P28223 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16166401 1.00 AKR1B1 (0.40) AKR1B1IDO1CBX7CDYL2CDYL
SCHEMBL16166210 0.92 KCNT1 (0.39) AKR1B1
SCHEMBL16166745 0.91 ELOVL6 (0.37) AKR1B1HTR2CHTR2B
SCHEMBL16175826 0.91 NPBWR1 (0.44) AKR1B1CBX7CDYLALDH1A1MEN1
SCHEMBL16166535 0.91 AKR1B1 (0.35) AKR1B1ALDH1A1POLBMEN1KMT2A
SCHEMBL16166284 0.89 AKR1B1 (0.36) AKR1B1HTR2CHTR2B
SCHEMBL16175837 0.89 NPBWR1 (0.44) CBX7CDYLALDH1A1MEN1KMT2A
SCHEMBL16166565 0.89 HTR2C (0.38) AKR1B1ALDH1A1TSHRHTR2C
SCHEMBL16166409 0.89 AKR1B1 (0.36) AKR1B1CBX7CDYL2CDYLCDY1; CDY1B
SCHEMBL16166339 0.89 IP6K1 (0.42) AKR1B1IDO1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014167528-A1 SPIROPYRAZOLOPYRIDINE DERIVATIVES AND USES THEREOF FOR THE TREATMENT OF VIRAL INFECTIONS NOVARTIS AG (CH) 2014-10-16 WO disclosed
WO-2014167528-A1 SPIROPYRAZOLOPYRIDINE DERIVATIVES AND USES THEREOF FOR THE TREATMENT OF VIRAL INFECTIONS NOVARTIS AG (CH) 2014-10-16 WO disclosed