SCHEMBL16166409

SCHEMBL16166409

O=C1C[C@]2(C(=O)Nc3ccc(Cl)cc32)c2cnn(Cc3ccc(OC(F)F)cc3)c2N1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 1/20 0.36
NPBWR1 P48145 1/20 0.32
P2RX3 P56373 3/20 0.32
DAO P14920 1/20 0.31
ADAMTS5 Q9UNA0 1/20 0.31
PSEN1 P49768 1/20 0.31
PSEN2 P49810 1/20 0.31
APH1B Q8WW43 1/20 0.31
NCSTN Q92542 1/20 0.31
APH1A Q96BI3 1/20 0.31
PSENEN Q9NZ42 1/20 0.31
MAOB P27338 1/20 0.31
CBX7 O95931 1/20 0.31
CDYL2 Q8N8U2 1/20 0.31
CDYL Q9Y232 1/20 0.31
CDY1; CDY1B Q9Y6F8 1/20 0.31
USP2 O75604 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
CPT1A P50416 1/20 0.31
CPT1B Q92523 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16166247 0.89 AKR1B1 (0.40) AKR1B1CBX7CDYL2CDYLCDY1; CDY1B
SCHEMBL16166401 0.89 AKR1B1 (0.40) AKR1B1CBX7CDYL2CDYLCDY1; CDY1B
SCHEMBL16175826 0.88 NPBWR1 (0.44) AKR1B1NPBWR1ADAMTS5CBX7CDYL
SCHEMBL16166565 0.88 HTR2C (0.38) AKR1B1
SCHEMBL16166745 0.85 ELOVL6 (0.37) AKR1B1NPBWR1
SCHEMBL16175837 0.85 NPBWR1 (0.44) NPBWR1ADAMTS5CBX7CDYL
SCHEMBL16166210 0.82 KCNT1 (0.39) AKR1B1
SCHEMBL16166284 0.81 AKR1B1 (0.36) AKR1B1NPBWR1P2RX3
SCHEMBL16166116 0.81 AKR1B1 (0.38) AKR1B1
SCHEMBL16166339 0.81 IP6K1 (0.42) AKR1B1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014167528-A1 SPIROPYRAZOLOPYRIDINE DERIVATIVES AND USES THEREOF FOR THE TREATMENT OF VIRAL INFECTIONS NOVARTIS AG (CH) 2014-10-16 WO disclosed
WO-2014167528-A1 SPIROPYRAZOLOPYRIDINE DERIVATIVES AND USES THEREOF FOR THE TREATMENT OF VIRAL INFECTIONS NOVARTIS AG (CH) 2014-10-16 WO disclosed