SCHEMBL16166295

SCHEMBL16166295

COc1cc(OC(OC)OC)c(CC=C(C)C)cc1CC=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 2/20 0.40
PTGES O14684 1/20 0.40
NFKB1 P19838 1/20 0.40
STAT3 P40763 1/20 0.40
NFKB2 Q00653 1/20 0.40
RELA Q04206 1/20 0.40
PPARG P37231 3/20 0.38
PTPN1 P18031 4/20 0.38
CYP19A1 P11511 3/20 0.36
MEN1 O00255 1/20 0.36
CES2 O00748 1/20 0.36
CES1 P23141 1/20 0.36
KMT2A Q03164 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
PDE4D Q08499 1/20 0.36
CYP3A4 P08684 1/20 0.36
IMPDH2 P12268 3/20 0.35
IMPDH1 P20839 2/20 0.35
AKR1C3 P42330 2/20 0.35
AKR1C2 P52895 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16166184 0.88 HTT (0.43) ALOX5PTGESNFKB1STAT3NFKB2
SCHEMBL16166638 0.74 ABCB1 (0.41) ALOX5PTGESNFKB1STAT3NFKB2
SCHEMBL16166508 0.72 AKR1C3 (0.41) ALOX5PTGESNFKB1STAT3NFKB2
SCHEMBL13403399 0.72 CYP3A4 (0.52) CYP19A1MEN1KMT2ATDP1CYP3A4
SCHEMBL21798818 0.72 TAAR1 (0.45) MEN1KMT2ATDP1CYP3A4IMPDH2
SCHEMBL16166422 0.70 TUBB1 (0.36) ALOX5PTGESNFKB1STAT3NFKB2
SCHEMBL16166393 0.69 ALOX5 (0.43) ALOX5PTGESPPARGPTPN1MEN1
SCHEMBL11155846 0.69 PTPN1 (0.48) ALOX5PTGESNFKB1STAT3NFKB2
SCHEMBL4268956 0.67 PTGS2 (0.41) ALOX5PTGESNFKB1STAT3NFKB2
SCHEMBL3303362 0.67 CYP19A1 (0.56) ALOX5PTGESNFKB1STAT3NFKB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2984072-A1 SYNTHETIC ANALOGUES OF XANTHOHUMOL Universita Di Pisa (IT) 2016-02-17 EP disclosed
WO-2014167481-A1 SYNTHETIC ANALOGUES OF XANTHOHUMOL UNIVERSITA' DI PISA (IT) 2014-10-16 WO disclosed