SCHEMBL16167673

SCHEMBL16167673

COc1cc(C(=O)NC(C)(C)C)ccc1S(=O)(=O)n1nc(-c2ccc(Cl)cc2)n(C2CC2)c1=O

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.38
NR1H4 Q96RI1 2/20 0.36
AVPR1A P37288 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
ALDH1A1 P00352 1/20 0.35
CNR1 P21554 3/20 0.35
CNR2 P34972 2/20 0.35
TACR2 P21452 1/20 0.35
TACR1 P25103 1/20 0.35
SCN9A Q15858 1/20 0.35
KMT2A Q03164 1/20 0.35
DDR1 Q08345 1/20 0.34
SMPD1 P17405 1/20 0.34
HTT P42858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16167675 0.87 ALDH1A1 (0.39) HSD11B1L3MBTL1AVPR1AALDH1A1KMT2A
SCHEMBL7911467 0.87 ALDH1A1 (0.39) HSD11B1L3MBTL1AVPR1ASMN1; SMN2ALDH1A1
SCHEMBL2511918 0.85 HSD11B1 (0.46) HSD11B1SMN1; SMN2ALDH1A1CNR1KMT2A
SCHEMBL7908197 0.84 ALDH1A1 (0.38) HSD11B1AVPR1AALDH1A1KMT2A
SCHEMBL7914828 0.84 AVPR1A (0.39) HSD11B1AVPR1ASMN1; SMN2ALDH1A1KMT2A
SCHEMBL16167674 0.83 AVPR1A (0.37) HSD11B1AVPR1ASMN1; SMN2ALDH1A1KMT2A
SCHEMBL7909318 0.83 AVPR1A (0.37) HSD11B1L3MBTL1AVPR1AALDH1A1CNR2
SCHEMBL7908194 0.83 KMT2A (0.38) HSD11B1AVPR1AALDH1A1CNR2KMT2A
SCHEMBL2500560 0.82 AVPR2 (0.41) HSD11B1AVPR1ASMN1; SMN2KMT2ASMPD1
SCHEMBL2513400 0.82 RXFP1 (0.37) HSD11B1L3MBTL1AVPR1ASMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8859601-B2 Substituted benzyl and phenylsulfonyl triazolones, and use thereof BAYER INTELLECTUAL PROPERTY GMBH (DE) 2014-10-14 US disclosed
US-8859601-B2 Substituted benzyl and phenylsulfonyl triazolones, and use thereof BAYER INTELLECTUAL PROPERTY GMBH (DE) 2014-10-14 US disclosed